SCHEMBL988515

SCHEMBL988515

COC(=O)COc1ccc(CCN(C)S(=O)(=O)c2ccc(F)cc2)cc1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 5/20 0.47
PDE4D Q08499 2/20 0.46
PTGER1 P34995 1/20 0.41
AR P10275 1/20 0.39
GPBAR1 Q8TDU6 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
CA9 Q16790 1/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MGAT3 Q09327 1/20 0.38
CYP3A4 P08684 1/20 0.37
SCN9A Q15858 1/20 0.37
MMP1 P03956 1/20 0.37
MMP9 P14780 1/20 0.37
MMP13 P45452 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL987716 0.92 PTGDR2 (0.57) PTGDR2PDE4DCA12CA1CA2
SCHEMBL2769871 0.83 PTGDR2 (0.58) PTGDR2CA12CA1CA2CA4
SCHEMBL12948817 0.82 PTGDR2 (0.45) PTGDR2ARGPBAR1ALDH1A1MAPT
SCHEMBL2770735 0.79 PTGDR2 (0.48) PTGDR2ARKDM4E
SCHEMBL2772208 0.77 PTGDR2 (0.62) PTGDR2CA12CA1CA2CA4
SCHEMBL2773541 0.77 PTGDR2 (0.58) PTGDR2CA12CA1CA2CA4
SCHEMBL988451 0.77 KEAP1 (0.46) PTGDR2PTGER1MMP1MMP9MMP13
SCHEMBL2773959 0.77 PTGDR2 (0.66) PTGDR2CA12CA1CA2CA4
SCHEMBL2771309 0.77 PTGDR2 (0.57) PTGDR2CA12CA1CA2CA4
SCHEMBL2770545 0.76 PTGDR2 (0.58) PTGDR2CA12CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002814-A2 BIARYL OXYACETIC ACID COMPOUNDS LIGAND PHARMACEUTICALS INC. (US) 2011-01-06 WO disclosed
WO-2010102154-A2 BIARYL OXYACETIC ACID COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-09-10 WO disclosed