SCHEMBL27710004

SCHEMBL27710004

CCOC(=O)CC1CCn2c1cc1c(C(C)C)nccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR Q13258 10/20 0.43
TBXA2R P21731 9/20 0.43
PTGER1 P34995 2/20 0.43
PTGER3 P43115 2/20 0.43
PTGER2 P43116 2/20 0.43
PTGDR2 Q9Y5Y4 2/20 0.43
PTGER4 P35408 1/20 0.43
PTGFR P43088 1/20 0.43
TLR8 Q9NR97 6/20 0.39
TLR7 Q9NYK1 6/20 0.39
TLR9 Q9NR96 4/20 0.39
NOS3 P29474 2/20 0.35
NOS1 P29475 2/20 0.35
NOS2 P35228 2/20 0.35
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA3 P34903 1/20 0.34
GABRA2 P47869 1/20 0.34
GABRB2 P47870 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2923853 0.86 PTGDR (0.53) PTGDRTBXA2RPTGER1PTGER3PTGER2
SCHEMBL13629399 0.82 PTGDR (0.39) PTGDRTBXA2RPTGER1PTGER3PTGER2
SCHEMBL13176192 0.81 PTGDR (0.43) PTGDRTBXA2RPTGER1PTGER3PTGER2
SCHEMBL27710012 0.80 PTGDR (0.39) PTGDRTBXA2RPTGER1PTGER3PTGER2
SCHEMBL2018070 0.78 GAA (0.37) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL2924355 0.77 PTGDR (0.39) PTGDRTBXA2RPTGER1PTGER3PTGER2
SCHEMBL2016666 0.77 S1PR1 (0.41) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL1255167 0.76 PTGDR (0.39) PTGDRTBXA2RPTGER1PTGER3PTGER2
SCHEMBL27631925 0.73 TBXA2R (0.44) PTGDRTBXA2R
SCHEMBL12320236 0.72 S1PR1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101189011-A Methods of treating atherosclerosis, lipid disorders and related conditions MERCK & CO INC (US) 2008-05-28 CN disclosed
CN-101056635-A Niacin receptor agonists, compositions containing such compounds and methods of treatment MERCK & CO INC (US) 2007-10-17 CN disclosed