SCHEMBL27714366

SCHEMBL27714366

N#CCc1ccc(Br)cc1CN

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CSNK2A1 P68400 4/20 0.47
CYP2A6 P11509 2/20 0.40
CCR5 P51681 1/20 0.37
PYCR1 P32322 2/20 0.32
HTR2A P28223 1/20 0.31
TRPM8 Q7Z2W7 1/20 0.31
BACE1 P56817 1/20 0.31
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30
NOS2 P35228 1/20 0.30
ESR1 P03372 1/20 0.30
ESR2 Q92731 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3390800 0.81 CYP2A6 (0.48) CYP2A6CCR5HTR2ATRPM8ALDH1A1
SCHEMBL1581581 0.81 CSNK2A1 (0.47) CSNK2A1PYCR1ALDH1A1HPGDNOS3
SCHEMBL5825 0.78 CSNK2A1 (0.49) CSNK2A1PYCR1
SCHEMBL29609415 0.78 CSNK2A1 (0.49) CSNK2A1PYCR1
SCHEMBL1758970 0.78 CSNK2A1 (0.49) CSNK2A1CYP2A6ALDH1A1
SCHEMBL11976907 0.78 CSNK2A1 (0.49) CSNK2A1CYP2A6PYCR1BACE1ALDH1A1
SCHEMBL20561966 0.78 CSNK2A1 (0.45) CSNK2A1PYCR1ALDH1A1HPGDNOS3
SCHEMBL28856582 0.78 CSNK2A1 (0.51) CSNK2A1CYP2A6PYCR1ALDH1A1HPGD
SCHEMBL2112768 0.78 CSNK2A1 (0.51) CSNK2A1CYP2A6PYCR1BACE1ALDH1A1
SCHEMBL4574084 0.77 CYP2A6 (0.47) CYP2A6HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101094827-B Benzene compound having two or more substituents DAIICHI SANKYO CO LTD 2012-06-13 CN disclosed
CN-101792436-A Benzimidazole derivatives used in the treatment of diseases associated with vanilloid receptor 1 ASTRAZENECA R & D SODERTALJE 2010-08-04 CN disclosed
CN-101522637-A Benzimidazole derivatives useful for the treatment of vanilloid receptor 1-related disorders ASTRAZENECA AB (SE) 2009-09-02 CN disclosed
CN-101094827-A Benzene compound having two or more substituents SANKYO CO (JP) 2007-12-26 CN disclosed