SCHEMBL27717137

SCHEMBL27717137

CC(N)Cc1c[nH]c2ccc([N+](=O)[O-])cc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.60
HTR2C P28335 4/20 0.60
HTR1A P08908 3/20 0.60
HTR2B P41595 3/20 0.60
HTR1B P28222 3/20 0.60
CYP2C19 P33261 2/20 0.60
HTR1D P28221 2/20 0.60
CYP1A2 P05177 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C9 P11712 1/20 0.60
NFKB1 P19838 1/20 0.60
PTPRA P18433 1/20 0.60
NQO2 P16083 1/20 0.56
ADRB1 P08588 1/20 0.55
ADRA2A P08913 1/20 0.55
SLC6A2 P23975 1/20 0.55
HTR1E P28566 1/20 0.55
SLC6A4 P31645 1/20 0.55
HTR7 P34969 1/20 0.55
HTR6 P50406 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16366296 0.90 PTPRA (0.73) HTR2AHTR2CHTR1AHTR2BHTR1B
SCHEMBL22316600 0.90 PTPRA (0.73) HTR2AHTR2CHTR1AHTR2BHTR1B
SCHEMBL10580344 0.86 NQO2 (0.56) CYP2C19PTPRANQO2SLC6A4PKM
SCHEMBL5115727 0.83 PTPRA (0.67) HTR2AHTR2CHTR1AHTR2BCYP2C19
SCHEMBL1580112 0.83 PTPRA (0.82) HTR2AHTR2CHTR1AHTR2BCYP2C19
SCHEMBL5115733 0.83 PTPRA (0.67) HTR2AHTR2CHTR1AHTR2BCYP2C19
SCHEMBL14032218 0.83 PTPRA (0.60) CYP2C19PTPRANQO2
SCHEMBL1580111 0.83 PTPRA (0.82) HTR2AHTR2CHTR1AHTR2BCYP2C19
SCHEMBL3294986 0.83 NQO2 (0.64) HTR2ANQO2SLC6A4PKMPKLR
SCHEMBL5773295 0.82 PTPRA (0.61) HTR2AHTR2CHTR1AHTR2BCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101272785-A Tetrahydro- beta-carbolin-sulfonamide derivatives as 5-HT6 ligands ESTEVE LABOR DR (ES) 2008-09-24 CN disclosed