SCHEMBL2772148

SCHEMBL2772148

Cc1cc(OCc2c(C)cnn2-c2c(Cl)cccc2Cl)ccc1CNCc1cccc(C(=O)O)c1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 10/20 0.51
NR1H4 Q96RI1 4/20 0.49
PPARA Q07869 1/20 0.45
NPC1 O15118 1/20 0.40
NR4A2 P43354 1/20 0.40
RAB9A P51151 1/20 0.40
BCL2 P10415 2/20 0.40
MCL1 Q07820 2/20 0.40
MEP1B Q16820 1/20 0.39
S1PR1 P21453 1/20 0.39
S1PR5 Q9H228 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2771623 0.92 NR1H4 (0.46) MRGPRX4NR1H4PPARANR4A2S1PR1
SCHEMBL2771176 0.91 NR1H4 (0.61) MRGPRX4NR1H4PPARA
SCHEMBL2773812 0.86 MRGPRX4 (0.48) MRGPRX4NR1H4PPARANPC1NR4A2
SCHEMBL3155316 0.86 MRGPRX4 (0.47) MRGPRX4NR1H4PPARANR4A2S1PR1
SCHEMBL2775204 0.85 MRGPRX4 (0.47) MRGPRX4NR1H4PPARANPC1NR4A2
SCHEMBL498490 0.85 NR1H4 (0.62) MRGPRX4NR1H4PPARA
SCHEMBL2773885 0.84 NR1H4 (0.59) MRGPRX4NR1H4PPARA
SCHEMBL2770433 0.84 MRGPRX4 (0.47) MRGPRX4NR1H4PPARANPC1NR4A2
SCHEMBL2770618 0.84 NR1H4 (0.58) MRGPRX4NR1H4PPARAS1PR1S1PR5
SCHEMBL2772150 0.83 MRGPRX4 (0.52) MRGPRX4NR1H4BCL2MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed