SCHEMBL2773885

SCHEMBL2773885

Cc1cc(OCc2c(C(C)C)cnn2-c2c(Cl)cccc2Cl)ccc1CNCCc1cccc(C(=O)O)c1

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 12/20 0.59
MRGPRX4 Q96LA9 6/20 0.45
PPARA Q07869 1/20 0.41
LIFR P42702 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2772215 0.93 NR1H4 (0.56) NR1H4MRGPRX4PPARALIFR
SCHEMBL2771176 0.93 NR1H4 (0.61) NR1H4MRGPRX4PPARALIFR
SCHEMBL2773434 0.89 NR1H4 (0.54) NR1H4MRGPRX4PPARA
SCHEMBL2770618 0.88 NR1H4 (0.58) NR1H4MRGPRX4PPARALIFR
SCHEMBL2772745 0.88 NR1H4 (0.53) NR1H4MRGPRX4PPARA
SCHEMBL2771368 0.87 NR1H4 (0.59) NR1H4MRGPRX4PPARALIFR
SCHEMBL2773673 0.86 NR1H4 (0.47) NR1H4PPARA
SCHEMBL2770317 0.86 NR1H4 (0.68) NR1H4MRGPRX4LIFR
SCHEMBL2771059 0.85 NR1H4 (0.57) NR1H4MRGPRX4PPARA
SCHEMBL2771221 0.85 NR1H4 (0.62) NR1H4MRGPRX4LIFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed