SCHEMBL27723391

SCHEMBL27723391

O=C(O)c1c[nH]c(-c2ccccc2F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 1/20 0.46
KDM4C Q9H3R0 1/20 0.46
KDM5B Q9UGL1 1/20 0.46
MAOA P21397 1/20 0.45
BLVRB P30043 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
TTR P02766 3/20 0.43
ACMSD Q8TDX5 1/20 0.43
NOTUM Q6P988 1/20 0.43
FFAR1 O14842 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
LDHA P00338 1/20 0.40
PTGER1 P34995 1/20 0.39
CSNK2A2 P19784 1/20 0.38
CSNK2B P67870 1/20 0.38
AXL P30530 1/20 0.38
DAO P14920 1/20 0.38
TSHR P16473 1/20 0.38
NAPRT Q6XQN6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28227720 0.87 TTR (0.44) KDM5AKDM4CKDM5BMAOABLVRB
SCHEMBL28654565 0.85 CDC7 (0.50) KDM5AKDM4CKDM5BFFAR1NPC1
SCHEMBL21666674 0.85 CDC7 (0.37) KDM5AKDM4CKDM5BMAOABLVRB
SCHEMBL21239294 0.83 KDM5A (0.35) KDM5AKDM4CKDM5BMAOABLVRB
SCHEMBL29815918 0.81 NPC1 (0.49) NPC1RAB9ATSHR
SCHEMBL31647020 0.81 GAA (0.46) HDAC6
SCHEMBL27743999 0.80 ALDH1A1 (0.47) TTRNOTUMFFAR1
SCHEMBL29237107 0.79 TDP1 (0.51) NPC1RAB9APTGER1TSHR
SCHEMBL30267515 0.78 JAK2 (0.49) RAB9ATSHR
SCHEMBL1156246 0.78 JAK2 (0.49) RAB9ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108148044-B Amide compound and method for preparing Vonoprazan fumarate from same 上海医药工业研究院 2024-05-14 CN claimed
CN-118978468-A Synthesis method of voronoi fumarate intermediate 武汉软件工程职业学院(武汉开放大学) 2024-11-19 CN disclosed
CN-108148044-B Amide compound and method for preparing Vonoprazan fumarate from same 上海医药工业研究院 2024-05-14 CN disclosed
CN-107915720-B Novel preparation method of Vonoprazan 常州市第四制药厂有限公司 2020-09-11 CN disclosed
CN-109843869-A 1- [(pyridin-3-yl-sulfonyl) -1H- pyrroles -3- base] methylamine derivative and its pharmaceutical composition and purposes 江苏吉贝尔药业股份有限公司 2019-06-04 CN disclosed
CN-101300229-B 1-heterocyclylsulfonyl, 2-aminomethyl, 5- (hetero-) aryl substituted 1-h-pyrrole derivatives as acid secretion inhibitors TAKEDA PHARMACEUTICAL 2011-10-05 CN disclosed
CN-101300229-A 1-heterocyclylsulfonyl, 2-aminomethyl, 5- (hetero-) aryl substituted 1-h-pyrrole derivatives as acid secretion inhibitors TAKEDA PHARMACEUTICAL (JP) 2008-11-05 CN disclosed