SCHEMBL27723722

SCHEMBL27723722

c1cc(-c2ccc(N3CCC4CCCCC4C3)cc2)ccn1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK13 O15264 1/20 0.53
MAPK12 P53778 1/20 0.53
MAPK11 Q15759 1/20 0.53
MAPK14 Q16539 1/20 0.53
IP6K1 Q92551 2/20 0.48
IP6K3 Q96PC2 2/20 0.48
IP6K2 Q9UHH9 1/20 0.48
IDO1 P14902 1/20 0.42
TDO2 P48775 1/20 0.42
CHKA P35790 1/20 0.42
HRH3 Q9Y5N1 2/20 0.38
CDK9 P50750 2/20 0.38
CHRNB2 P17787 2/20 0.38
CHRNB4 P30926 2/20 0.38
CHRNA3 P32297 2/20 0.38
CHRNA4 P43681 2/20 0.38
CYP17A1 P05093 3/20 0.37
CYP21A2 P08686 3/20 0.37
CYP11B1 P15538 2/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6607442 0.77 MAPT (0.48) MAPK13MAPK12MAPK11MAPK14IP6K1
SCHEMBL6606401 0.77 MAPT (0.48) MAPK13MAPK12MAPK11MAPK14IP6K1
SCHEMBL6712762 0.77 MAPT (0.48) MAPK13MAPK12MAPK11MAPK14IP6K1
SCHEMBL31175194 0.76 NOTUM (0.51) IP6K1IP6K3IP6K2TDO2HRH3
SCHEMBL15101965 0.76 CHKA (0.54) MAPK13MAPK12MAPK11MAPK14IP6K1
SCHEMBL25506010 0.76 CHKA (0.54) MAPK13MAPK12MAPK11MAPK14IP6K1
SCHEMBL28281275 0.74 CHKA (0.75) CHKACDK9CYP3A4MELK
SCHEMBL15496950 0.73 GPR119 (0.48) IP6K1IP6K3IP6K2HRH3CHRNB2
SCHEMBL38662172 0.72 CHKA (0.50) MAPK13MAPK12MAPK11MAPK14CHKA
SCHEMBL28229454 0.72 CHKA (0.42) IDO1TDO2CHKACYP17A1CYP21A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101253152-A Amide derivatives as ROCK inhibitors ASTELLAS PHARMA INC (JP) 2008-08-27 CN disclosed