SCHEMBL27723934

SCHEMBL27723934

CCCCOC(=O)Nc1cccnc1C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.55
CYP1A2 P05177 2/20 0.55
CYP2C19 P33261 2/20 0.55
GAA P10253 3/20 0.51
PTPN1 P18031 1/20 0.51
L3MBTL1 Q9Y468 3/20 0.50
BRD4 O60885 1/20 0.50
ALDH1A1 P00352 6/20 0.49
RAB9A P51151 6/20 0.48
NPC1 O15118 5/20 0.48
TSHR P16473 1/20 0.46
HPGD P15428 4/20 0.46
KDM4E B2RXH2 3/20 0.46
LMNA P02545 1/20 0.46
CSNK2A2 P19784 1/20 0.46
CSNK2A1 P68400 1/20 0.46
ALOX15 P16050 1/20 0.45
NFKB1 P19838 1/20 0.45
STAT1 P42224 1/20 0.45
NFKB2 Q00653 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4443244 0.87 BRD4 (0.68) SMN1; SMN2CYP1A2CYP2C19GAAPTPN1
SCHEMBL5572207 0.81 SMN1; SMN2 (0.54) SMN1; SMN2CYP1A2CYP2C19GAAL3MBTL1
SCHEMBL8192523 0.81 SMN1; SMN2 (0.54) SMN1; SMN2CYP1A2CYP2C19GAAL3MBTL1
SCHEMBL8203991 0.81 SMN1; SMN2 (0.57) SMN1; SMN2CYP1A2CYP2C19GAAPTPN1
SCHEMBL31082406 0.80 KDM4E (0.52) CYP1A2GAAPTPN1L3MBTL1BRD4
SCHEMBL14214178 0.80 MEN1 (0.59) SMN1; SMN2CYP1A2CYP2C19GAAL3MBTL1
SCHEMBL3655453 0.79 SMN1; SMN2 (0.52) SMN1; SMN2CYP1A2CYP2C19GAAPTPN1
SCHEMBL2320061 0.78 SMN1; SMN2 (0.77) SMN1; SMN2CYP1A2CYP2C19L3MBTL1ALDH1A1
SCHEMBL15348811 0.77 GAA (0.64) SMN1; SMN2CYP1A2CYP2C19GAAL3MBTL1
SCHEMBL8200993 0.76 SMN1; SMN2 (0.52) SMN1; SMN2CYP1A2CYP2C19GAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101189243-A Substituted heterocycles and their use as CHK1, PDK1 and PAK inhibitors ASTRAZENECA AB (SE) 2008-05-28 CN disclosed