SCHEMBL27734733

SCHEMBL27734733

Cc1c(Oc2ccc(CCn3ccnc3)cc2F)ncnc1OC1CCN(C(=O)O)CC1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 16/20 0.49
CYP2C9 P11712 1/20 0.49
PIK3CD O00329 3/20 0.42
NTRK1 P04629 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL390104 0.90 GPR119 (0.64) GPR119CYP2C9
SCHEMBL3168629 0.86 GPR119 (0.51) GPR119CYP2C9PIK3CD
SCHEMBL27734761 0.86 GPR119 (0.49) GPR119CYP2C9PIK3CD
SCHEMBL1071546 0.83 GPR119 (0.56) GPR119CYP2C9PIK3CDNTRK1
SCHEMBL27734782 0.81 GPR119 (0.48) GPR119CYP2C9PIK3CD
SCHEMBL27755351 0.80 GPR119 (0.51) GPR119CYP2C9PIK3CD
SCHEMBL1068483 0.79 GPR119 (0.52) GPR119CYP2C9PIK3CDNTRK1
SCHEMBL27734866 0.77 GPR119 (0.50) GPR119CYP2C9PIK3CDNTRK1
SCHEMBL389602 0.76 GPR119 (0.64) GPR119CYP2C9
SCHEMBL27734759 0.76 GPR119 (0.56) GPR119CYP2C9PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101420941-A Use of GPR119 receptor agonists for increasing bone mass and for treating osteoporosis, and related combination therapies ARENA PHARM INC (US) 2009-04-29 CN disclosed
CN-101332303-A Combination therapy for the treatment of diabetes and conditions related thereto and for the treatment of conditions ameliorated by increasing a blood glp-1 level ARENA PHARM INC (US) 2008-12-31 CN disclosed