SCHEMBL2773539

SCHEMBL2773539

Cc1cc(OCc2c(C(C)C)cnn2-c2c(Cl)cccc2Cl)ccc1-c1cc2cccc(C(=O)O)c2s1

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 19/20 0.54
NR1I2 O75469 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
MRGPRX4 Q96LA9 1/20 0.34
VDR P11473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2770454 0.85 NR1H4 (0.59) NR1H4MRGPRX4VDR
SCHEMBL2770414 0.85 NR1H4 (0.57) NR1H4MRGPRX4
SCHEMBL2773272 0.83 NR1H4 (0.57) NR1H4
SCHEMBL2774467 0.83 NR1H4 (0.57) NR1H4
SCHEMBL2770495 0.83 NR1H4 (0.67) NR1H4MRGPRX4VDR
SCHEMBL2772857 0.83 NR1H4 (0.55) NR1H4MRGPRX4VDR
SCHEMBL2771077 0.83 NR1H4 (0.55) NR1H4
SCHEMBL2770807 0.83 NR1H4 (0.58) NR1H4MRGPRX4VDR
SCHEMBL2770415 0.82 NR1H4 (0.54) NR1H4MRGPRX4VDR
SCHEMBL2771697 0.81 NR1H4 (0.63) NR1H4MRGPRX4VDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed