SCHEMBL2772857

SCHEMBL2772857

Cc1cc(OCc2c(C(C)C)cnn2-c2c(Cl)cccc2Cl)ccc1-c1nc(C)c(C(=O)O)s1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 9/20 0.55
TARBP2 Q15633 2/20 0.40
FFAR2 O15552 1/20 0.39
NPSR1 Q6W5P4 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.35
VDR P11473 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
POLB P06746 1/20 0.34
RAB9A P51151 1/20 0.34
PPARD Q03181 2/20 0.34
PDE5A O76074 1/20 0.34
PDE1A P54750 1/20 0.34
PDE1B Q01064 1/20 0.34
PDE1C Q14123 1/20 0.34
PPARA Q07869 1/20 0.34
ABCC4 O15439 1/20 0.34
ABCB11 O95342 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2774019 0.89 NR1H4 (0.54) NR1H4TARBP2SMN1; SMN2KDM4ENPC1
SCHEMBL2770414 0.85 NR1H4 (0.57) NR1H4MRGPRX4SMN1; SMN2KDM4ENPC1
SCHEMBL2770495 0.84 NR1H4 (0.67) NR1H4MRGPRX4VDR
SCHEMBL2770807 0.84 NR1H4 (0.58) NR1H4MRGPRX4VDR
SCHEMBL2773539 0.83 NR1H4 (0.54) NR1H4MRGPRX4VDR
SCHEMBL2771697 0.83 NR1H4 (0.63) NR1H4MRGPRX4VDR
SCHEMBL2770454 0.82 NR1H4 (0.59) NR1H4MRGPRX4VDR
SCHEMBL2772894 0.82 NR1H4 (0.67) NR1H4MRGPRX4
SCHEMBL2772951 0.82 NR1H4 (0.37) NR1H4TARBP2NPSR1RXFP1PPARD
SCHEMBL2770415 0.82 NR1H4 (0.54) NR1H4MRGPRX4VDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed