SCHEMBL2773595

SCHEMBL2773595

COC(=O)c1ccc(C#N)cc1F.COC(=O)c1ccc(C(N)=NO)cc1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.41
GAA P10253 2/20 0.41
TRPA1 O75762 1/20 0.41
MAP2K1 Q02750 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
ALDH1A1 P00352 3/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
MAPT P10636 3/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
POLB P06746 2/20 0.40
KDM4E B2RXH2 1/20 0.40
GLA P06280 1/20 0.40
HPGD P15428 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
ATM Q13315 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL406865 0.90 KDM4E (0.47) SMN1; SMN2GAAALDH1A1NPC1RAB9A
SCHEMBL406864 0.90 KDM4E (0.47) SMN1; SMN2GAAALDH1A1NPC1RAB9A
SCHEMBL8401255 0.90 KDM4E (0.47) SMN1; SMN2GAAALDH1A1NPC1RAB9A
SCHEMBL2773888 0.84 MRGPRX4 (0.43) SMN1; SMN2GAAALDH1A1NPC1RAB9A
SCHEMBL409948 0.84 MEN1 (0.50) SMN1; SMN2GAAMAP2K1CYP11B1CYP11B2
SCHEMBL536199 0.82 MEN1 (0.46) SMN1; SMN2GAATRPA1MAP2K1CYP11B1
SCHEMBL9968898 0.79 KDM4E (0.51) SMN1; SMN2GAAALDH1A1MAPTKMT2A
SCHEMBL2776989 0.79 KDM4E (0.51) SMN1; SMN2GAAALDH1A1MAPTKMT2A
SCHEMBL9968900 0.79 RECQL (0.45) SMN1; SMN2GAAALDH1A1NPC1RAB9A
SCHEMBL2776991 0.79 KDM4E (0.51) SMN1; SMN2GAAALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2193125-A2 OXADIAZOLE DERIVATIVES Merck Serono S.A. (CH) 2010-06-09 EP disclosed
WO-2009043889-A2 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2009-04-09 WO disclosed