SCHEMBL27736552

SCHEMBL27736552

CC(C)(C)OOC(=O)c1ccc(NC(=O)c2ccc3ccn(S(=O)(=O)c4cccc(Cl)c4)c3c2)cc1

nearest known ligand 0.73

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CPT1A P50416 11/20 0.73
CPT1B Q92523 9/20 0.73
CPT2 P23786 7/20 0.73
PPARG P37231 7/20 0.50
PPARD Q03181 7/20 0.50
PPARA Q07869 7/20 0.50
STAT3 P40763 1/20 0.45
CYP3A4 P08684 1/20 0.45
HTR6 P50406 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3577725 0.91 CPT1A (0.75) CPT1ACPT1BCPT2PPARGPPARD
SCHEMBL27715639 0.86 CPT1A (0.72) CPT1ACPT1BCPT2PPARGPPARD
SCHEMBL3572875 0.84 CPT1A (1.00) CPT1ACPT1BCPT2PPARGPPARD
SCHEMBL2906020 0.84 CPT1A (0.77) CPT1ACPT1BCPT2PPARGPPARD
SCHEMBL27877814 0.82 CPT1A (0.71) CPT1ACPT1BCPT2PPARGPPARD
SCHEMBL2898335 0.80 CPT1A (1.00) CPT1ACPT1BCPT2PPARGPPARD
SCHEMBL3568174 0.77 CPT1A (0.75) CPT1ACPT1BCPT2PPARGPPARD
SCHEMBL27736550 0.76 CPT1A (0.56) CPT1ACPT1BCPT2PPARGPPARD
SCHEMBL27751900 0.76 CPT1A (0.75) CPT1ACPT1BCPT2PPARG
SCHEMBL3576367 0.72 CPT1A (0.76) CPT1ACPT1BCPT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101263116-B Novel heterobicyclic derivatives useful as liver carnitine palmitoyl transferase inhibitors HOFFMAN-LA ROCHE LTD. (CH) 2011-12-07 CN disclosed
CN-101263116-A Novel heterobicyclic derivatives useful as liver carnitine palmitoyl transferase inhibitors HOFFMANN LA ROCHE (CH) 2008-09-10 CN disclosed