SCHEMBL27737390

SCHEMBL27737390

CC(C)(C)C(=O)ON1CC=C(c2ccc(-c3cnc(Nc4cccc(Cl)c4)o3)cc2)CC1

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.63
SIRT7 Q9NRC8 1/20 0.44
VCP P55072 3/20 0.42
KDR P35968 8/20 0.42
FLT1 P17948 7/20 0.42
FLT4 P35916 7/20 0.42
TRPV1 Q8NER1 3/20 0.37
IMPDH2 P12268 1/20 0.36
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL180759 0.85 DGAT1 (0.70) DGAT1SIRT7VCPKDRFLT1
SCHEMBL180635 0.81 DGAT1 (0.58) DGAT1SIRT7VCPKDRFLT1
SCHEMBL180813 0.81 DGAT1 (0.79) DGAT1SIRT7VCPKDRFLT1
SCHEMBL181174 0.80 DGAT1 (0.77) DGAT1SIRT7VCPKDRFLT1
SCHEMBL180683 0.79 DGAT1 (0.70) DGAT1SIRT7VCPKDRFLT1
SCHEMBL180970 0.78 DGAT1 (0.65) DGAT1SIRT7VCPKDRFLT1
SCHEMBL180428 0.77 DGAT1 (1.00) DGAT1SIRT7VCPKDRFLT1
SCHEMBL180799 0.77 DGAT1 (0.72) DGAT1SIRT7VCPKDRFLT1
SCHEMBL27488925 0.74 PPARG (0.46) LMNAMAPTHTTNPSR1
Tert-Butyl Formate SCHEMBL27737391 0.72 DGAT1 (0.49) DGAT1SIRT7VCPKDRFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103288721-A (4-(4-[6-(trifluoromethyl-pyridin-3-ylamino)-n-containing-heteroaryl]-phenyl)-cyclohexyl)-acetic acid derivatives and pharmaceutical uses thereof NOVARTIS AG 2013-09-11 CN disclosed
CN-101415683-B Novel compounds NOVARTIS AG 2013-07-17 CN disclosed
CN-103086981-A New compounds NOVARTIS AG 2013-05-08 CN disclosed
CN-101415683-A Novel compounds NOVARTIS AG (CH) 2009-04-22 CN disclosed