SCHEMBL2773673

SCHEMBL2773673

CCCCOc1ccc(CCNCc2ccc(OCc3c(C(C)C)cnn3-c3c(Cl)cccc3Cl)cc2C)cc1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 7/20 0.47
CYP2D6 P10635 4/20 0.34
KCNH2 Q12809 1/20 0.34
PPARD Q03181 5/20 0.33
PDGFRA P16234 1/20 0.33
S1PR1 P21453 1/20 0.33
ROCK1 Q13464 1/20 0.33
S1PR5 Q9H228 1/20 0.33
PPARA Q07869 3/20 0.33
PPARG P37231 3/20 0.33
ADRB1 P08588 1/20 0.33
ADRB3 P13945 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2770409 0.94 NR1H4 (0.49) NR1H4PPARDPDGFRAS1PR1ROCK1
SCHEMBL2771506 0.89 NR1H4 (0.49) NR1H4PPARDPDGFRAS1PR1ROCK1
SCHEMBL2772215 0.87 NR1H4 (0.56) NR1H4PPARDPDGFRAS1PR1ROCK1
SCHEMBL2773885 0.86 NR1H4 (0.59) NR1H4PPARA
SCHEMBL2773434 0.85 NR1H4 (0.54) NR1H4PDGFRAS1PR1ROCK1S1PR5
SCHEMBL2773675 0.85 NR1H4 (0.48) NR1H4PPARDPPARAPPARG
SCHEMBL2771518 0.84 NR1H4 (0.50) NR1H4
SCHEMBL2772745 0.84 NR1H4 (0.53) NR1H4PPARDPDGFRAS1PR1ROCK1
SCHEMBL2772157 0.83 NR1H4 (0.53) NR1H4PPARDPPARAPPARG
SCHEMBL2773708 0.83 NR1H4 (0.53) NR1H4PPARDPPARAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed