SCHEMBL27740959

SCHEMBL27740959

COc1c(C(F)(F)F)nnn1-c1ccccc1OC(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 5/20 0.40
HSD11B1 P28845 1/20 0.39
HCAR1 Q9BXC0 4/20 0.37
SCN9A Q15858 2/20 0.36
ALDH1A1 P00352 2/20 0.36
NR1I2 O75469 1/20 0.35
P2RX7 Q99572 2/20 0.35
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL498054 0.77 KCNN4 (0.42) KCNN4HSD11B1HCAR1SCN9AALDH1A1
SCHEMBL498090 0.73 SLC5A1 (0.46) KCNN4HCAR1SCN9AALDH1A1HSD17B10
SCHEMBL28460135 0.69 KCNN4 (0.52) KCNN4HSD11B1HCAR1SCN9AALDH1A1
SCHEMBL1493544 0.69 KCNN4 (0.52) KCNN4HSD11B1HCAR1SCN9AALDH1A1
SCHEMBL497639 0.67 KCNN4 (0.40) KCNN4HSD11B1HCAR1SCN9AALDH1A1
SCHEMBL14996565 0.67 MAPT (0.47) KCNN4HSD11B1HCAR1SCN9AALDH1A1
SCHEMBL28188336 0.67 KCNN4 (0.47) KCNN4HSD11B1HCAR1SCN9AALDH1A1
SCHEMBL4205517 0.66 KCNN4 (0.56) KCNN4ALDH1A1TSHRHTTHSD17B10
SCHEMBL12859430 0.65 SCN9A (0.43) KCNN4HSD11B1HCAR1SCN9AALDH1A1
SCHEMBL5906114 0.65 HCAR1 (0.47) KCNN4HCAR1SCN9AP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101448798-A Compounds and methods for modulating FXR LILLY CO ELI (US) 2009-06-03 CN disclosed