SCHEMBL27745238

SCHEMBL27745238

CCOC(=O)CCCC(=O)c1ccc(F)c(F)c1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.46
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
CYP4F2 P78329 3/20 0.41
CYP4A11 Q02928 3/20 0.41
NPC1 O15118 1/20 0.40
LMNA P02545 2/20 0.39
NR1I2 O75469 1/20 0.39
PGR P06401 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
PTGS2 P35354 1/20 0.39
PDE4D Q08499 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TSHR P16473 1/20 0.39
USP2 O75604 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TNF P01375 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL312535 0.84 CES2 (0.47) CYP1A2CES2CES1NPC1LMNA
SCHEMBL1361469 0.80 CYP4F2 (0.50) CYP1A2CYP4F2CYP4A11TNFALDH1A1
SCHEMBL1958113 0.79 TSHR (0.57) CES2CES1LMNATSHRHSD17B10
SCHEMBL8585798 0.78 CYP4F2 (0.57) CYP1A2CYP4F2CYP4A11NPC1L3MBTL1
SCHEMBL6623875 0.77 CES2 (0.53) CYP1A2CES2CES1NPC1LMNA
SCHEMBL29775615 0.76 CES2 (0.44) CYP1A2CES2CES1NPC1LMNA
SCHEMBL21047313 0.76 CES2 (0.44) CYP1A2CES2CES1NPC1LMNA
SCHEMBL2743554 0.75 NPC1 (0.68) CYP1A2NPC1LMNAL3MBTL1TSHR
SCHEMBL7860050 0.75 CYP4F2 (0.54) CYP1A2CYP4F2CYP4A11LMNAALDH1A1
SCHEMBL2373430 0.75 CES2 (0.59) CES2CES1L3MBTL1TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101312972-B Bicyclic cinnamide compound EISAI R&D MAN CO LTD 2012-06-20 CN disclosed
CN-101312972-A Bicyclic cinnamide compound EISAI R&D MAN CO LTD (JP) 2008-11-26 CN disclosed