SCHEMBL27745889

SCHEMBL27745889

Cc1c(C)c(-c2ccc(F)cc2Cl)c(C(=O)O)c(-c2nccs2)c1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
DHODH Q02127 5/20 0.38
CDC7 O00311 1/20 0.38
DBF4 Q9UBU7 1/20 0.38
EIF4E P06730 1/20 0.37
F2RL1 P55085 1/20 0.36
TRPM4 Q8TD43 1/20 0.35
P2RX7 Q99572 1/20 0.35
KCNH2 Q12809 1/20 0.34
ECE1 P42892 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ROS1 P08922 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27725074 0.89 HDAC3 (0.41) HDAC3HDAC1HDAC6DHODHCDC7
SCHEMBL27748447 0.87 KCNH2 (0.37) HDAC3HDAC1HDAC6DHODHF2RL1
SCHEMBL19259491 0.79 HDAC3 (0.43) HDAC3HDAC1HDAC6DHODHCDC7
SCHEMBL27727426 0.76 KCNH2 (0.37) HDAC3HDAC1HDAC6DHODHF2RL1
SCHEMBL27745887 0.76 HDAC3 (0.40) HDAC3HDAC1HDAC6CDC7DBF4
SCHEMBL27725072 0.74 CDC7 (0.47) HDAC3HDAC1HDAC6CDC7DBF4
SCHEMBL405716 0.73 EIF4E (0.44) HDAC3HDAC1HDAC6EIF4EF2RL1
SCHEMBL16237487 0.72 HDAC3 (0.43) HDAC3HDAC1HDAC6DHODHCDC7
SCHEMBL15515454 0.70 CDC7 (0.43) HDAC3HDAC1HDAC6DHODHCDC7
SCHEMBL27690481 0.69 EIF4E (0.42) DHODHCDC7DBF4EIF4EP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101328170-B Fluorophenyl-substituted thiazole dihydropyrimidine ZHANG ZHONGNENG 2011-09-14 CN disclosed
CN-101328168-B Diethylcarbamyl-substituted thiazole dihydropyrimidine ZHANG ZHONGNENG 2011-09-07 CN disclosed
CN-101328168-A Diethylcarbamyl-substituted thiazole dihydropyrimidine ZHANG ZHONGNENG (CN) 2008-12-24 CN disclosed
CN-101328170-A Fluorophenyl-substituted thiazole dihydropyrimidine ZHANG ZHONGNENG (CN) 2008-12-24 CN disclosed