SCHEMBL27746307

SCHEMBL27746307

CN(C)C=CC(=O)C(=O)C(=O)C=CN(C)C

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.48
HTT P42858 3/20 0.43
RECQL P46063 2/20 0.41
MAPT P10636 7/20 0.39
RAB9A P51151 5/20 0.39
LMNA P02545 4/20 0.39
HPGD P15428 3/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C19 P33261 2/20 0.39
ALOX12 P18054 1/20 0.39
ALDH1A1 P00352 8/20 0.36
POLB P06746 3/20 0.36
KMT2A Q03164 3/20 0.35
NPC1 O15118 3/20 0.35
KDM4E B2RXH2 2/20 0.35
GAA P10253 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13887197 0.80 TDP1 (0.46) TDP1HTTRECQLMAPTRAB9A
SCHEMBL932497 0.80 TDP1 (0.46) TDP1HTTRECQLMAPTRAB9A
SCHEMBL932496 0.80 TDP1 (0.46) TDP1HTTRECQLMAPTRAB9A
SCHEMBL10418299 0.80 TDP1 (0.46) TDP1HTTRECQLMAPTRAB9A
SCHEMBL6822957 0.78 TDP1 (0.50) TDP1HTTRECQLMAPTRAB9A
SCHEMBL6822956 0.78 TDP1 (0.50) TDP1HTTRECQLMAPTRAB9A
SCHEMBL7345258 0.75 TDP1 (0.52) TDP1HTTRECQLMAPTRAB9A
SCHEMBL7345262 0.75 TDP1 (0.52) TDP1HTTRECQLMAPTRAB9A
SCHEMBL4378106 0.74 MAPT (0.48) TDP1HTTRECQLMAPTRAB9A
SCHEMBL4378103 0.74 MAPT (0.48) TDP1HTTRECQLMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101754968-A Substituted imidazopyridazines as PI3K lipid kinase inhibitors NOVARTIS AG 2010-06-23 CN disclosed
CN-101321763-A Pyrazolo [1,5-a] pyrimidines as protein kinase inhibitors SCHERING CORP (US) 2008-12-10 CN disclosed