SCHEMBL27747341

SCHEMBL27747341

CC(=S)CCCc1nnc(C(N)=O)c2sc(-c3ccc(Cl)cc3)cc12

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 13/20 0.47
IKBKB O14920 2/20 0.39
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
POLB P06746 1/20 0.38
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
RAB9A P51151 1/20 0.34
GFER P55789 1/20 0.34
KMT2A Q03164 1/20 0.34
MAP3K8 P41279 2/20 0.34
STK17B O94768 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27768306 0.90 IKBKB (0.39) CHEK1IKBKBMAPTKDM4EMEN1
SCHEMBL27747338 0.90 CHEK1 (0.37) CHEK1MAPTPOLBKDM4EMEN1
SCHEMBL28776699 0.82 CHEK1 (0.34) CHEK1ALDH1A1MAPTPOLBKDM4E
SCHEMBL12922001 0.79 CHEK1 (0.48) CHEK1IKBKBMAP3K8STK17B
SCHEMBL8827896 0.78 CHEK1 (0.47) CHEK1IKBKBALDH1A1MAPTPOLB
SCHEMBL14997868 0.77 CHEK1 (0.45) CHEK1IKBKBALDH1A1MAPTPOLB
SCHEMBL12922023 0.76 CHEK1 (0.57) CHEK1IKBKBALDH1A1MAPTKDM4E
SCHEMBL29900031 0.76 CHEK1 (0.46) CHEK1IKBKBALDH1A1KDM4E
SCHEMBL12921998 0.76 CHEK1 (0.46) CHEK1IKBKBALDH1A1KDM4E
SCHEMBL12922015 0.76 CHEK1 (0.56) CHEK1IKBKBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101481380-A Thiofuran pyridazine compound, preparation thereof, pharmaceutical composition and uses thereof ZHEJIANG MEDICINE CO LTD (CN) 2009-07-15 CN claimed
CN-101481380-A Thiofuran pyridazine compound, preparation thereof, pharmaceutical composition and uses thereof ZHEJIANG MEDICINE CO LTD (CN) 2009-07-15 CN disclosed