SCHEMBL27747802

SCHEMBL27747802

Cc1c(Oc2ccc(OC3CCOCC3)cc2F)ncnc1OC1CCN(C(=O)O)CC1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 17/20 0.55
CYP2C9 P11712 1/20 0.55
PIK3CD O00329 2/20 0.46
ACACB O00763 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL386518 0.89 GPR119 (0.71) GPR119CYP2C9
SCHEMBL1068483 0.84 GPR119 (0.52) GPR119CYP2C9PIK3CD
SCHEMBL27755093 0.84 GPR119 (0.53) GPR119CYP2C9PIK3CDACACB
SCHEMBL27734703 0.84 GPR119 (0.53) GPR119CYP2C9PIK3CD
SCHEMBL3160437 0.84 GPR119 (0.56) GPR119CYP2C9ACACB
SCHEMBL27734793 0.83 GPR119 (0.53) GPR119CYP2C9PIK3CD
SCHEMBL27747878 0.82 GPR119 (0.52) GPR119CYP2C9PIK3CD
SCHEMBL1071546 0.81 GPR119 (0.56) GPR119CYP2C9PIK3CD
SCHEMBL27734759 0.81 GPR119 (0.56) GPR119CYP2C9PIK3CD
SCHEMBL2786447 0.81 GPR119 (0.79) GPR119CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101420941-A Use of GPR119 receptor agonists for increasing bone mass and for treating osteoporosis, and related combination therapies ARENA PHARM INC (US) 2009-04-29 CN disclosed