SCHEMBL27747879

SCHEMBL27747879

CC(C)OC(=O)N1CCC(Oc2ncnc3c2cnn3-c2ccc(S(=O)(=O)NF)cc2)CC1

nearest known ligand 0.82

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 20/20 0.82
CYP2C9 P11712 3/20 0.68
KCNH2 Q12809 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL388759 0.90 GPR119 (1.00) GPR119CYP2C9KCNH2
SCHEMBL390682 0.86 GPR119 (0.79) GPR119CYP2C9KCNH2
SCHEMBL388204 0.86 GPR119 (0.79) GPR119CYP2C9KCNH2
SCHEMBL386623 0.85 GPR119 (0.76) GPR119CYP2C9KCNH2
SCHEMBL391165 0.84 GPR119 (0.71) GPR119CYP2C9KCNH2
SCHEMBL388652 0.83 GPR119 (0.76) GPR119CYP2C9KCNH2
SCHEMBL10170747 0.83 GPR119 (0.86) GPR119CYP2C9KCNH2
SCHEMBL390792 0.83 GPR119 (0.69) GPR119CYP2C9KCNH2
SCHEMBL389847 0.81 GPR119 (0.84) GPR119CYP2C9KCNH2
SCHEMBL391161 0.81 GPR119 (0.83) GPR119CYP2C9KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101420941-A Use of GPR119 receptor agonists for increasing bone mass and for treating osteoporosis, and related combination therapies ARENA PHARM INC (US) 2009-04-29 CN disclosed