SCHEMBL2774798

SCHEMBL2774798

CC(C)[C@H](NC(=O)O)C(=O)N1CCC(OC2CCCCC2)CC1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45
CCR1 P32246 13/20 0.43
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
KMT2A Q03164 1/20 0.42
HPGD P15428 1/20 0.40
KCNH2 Q12809 1/20 0.40
POLB P06746 1/20 0.38
DPP4 P27487 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2774643 0.79 CCR1 (0.45) CYP3A4CYP2C19CCR1KCNH2
SCHEMBL25320081 0.78 CYP3A4 (0.46) CYP3A4CYP2C19CCR1LMNAKMT2A
SCHEMBL12632401 0.78 CYP3A4 (0.46) CYP3A4CYP2C19CCR1LMNAKMT2A
SCHEMBL15458220 0.78 CYP3A4 (0.46) CYP3A4CYP2C19CCR1LMNAKMT2A
Hydrochloric Acid SCHEMBL2774871 0.75 DPP4 (0.42) DPP4
SCHEMBL2778524 0.75 CCR1 (0.45) CCR1KMT2AKCNH2
SCHEMBL2775929 0.74 KMT2A (0.45) CCR1LMNATSHRKMT2AKCNH2
SCHEMBL2775987 0.74 ACACB (0.42) CYP3A4CYP2C19CCR1POLB
SCHEMBL2776114 0.74 ACACB (0.46) CYP3A4CYP2C19CCR1LMNATSHR
SCHEMBL2775803 0.74 CCR1 (0.55) CCR1LMNATSHRKMT2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2258697-A1 HYDROXYQUINOXALINECARBOXAMIDE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2010-12-08 EP disclosed