SCHEMBL2774643

SCHEMBL2774643

CC(C)[C@H](NC(=O)O)C(=O)N1CCC(O)CC1

nearest known ligand 0.45

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 17/20 0.45
KCNH2 Q12809 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2773444 0.83 ITGB3 (0.41)
SCHEMBL12632401 0.82 CYP3A4 (0.46) CCR1KCNH2CYP3A4CYP2C19
SCHEMBL25320081 0.82 CYP3A4 (0.46) CCR1KCNH2CYP3A4CYP2C19
SCHEMBL15458220 0.82 CYP3A4 (0.46) CCR1KCNH2CYP3A4CYP2C19
SCHEMBL2774798 0.79 CYP3A4 (0.45) CCR1KCNH2CYP3A4CYP2C19
SCHEMBL2775499 0.79 KMT2A (0.55) CCR1CYP3A4CYP2C19
SCHEMBL14779934 0.78 SMN1; SMN2 (0.50) CCR1CYP3A4CYP2C19
SCHEMBL2776192 0.75 CCR1 (0.46) CCR1
SCHEMBL21531141 0.75 CCR1 (0.80) CCR1KCNH2
SCHEMBL17527163 0.74 DPP4 (0.52) KCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2258697-A1 HYDROXYQUINOXALINECARBOXAMIDE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2010-12-08 EP disclosed