SCHEMBL277482

SCHEMBL277482

C1CCN(CN2CCCC2)C1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.47
HRH3 Q9Y5N1 3/20 0.44
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
CARM1 Q86X55 1/20 0.38
PRMT6 Q96LA8 1/20 0.38
PRMT8 Q9NR22 1/20 0.38
CHRM5 P08912 1/20 0.38
ADRA2C P18825 1/20 0.38
MAPT P10636 4/20 0.36
ATM Q13315 1/20 0.36
TSHR P16473 1/20 0.36
GAA P10253 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.33
HRH4 Q9H3N8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1799442 0.96 HRH3 (0.50) LMNAHRH3KMT2AMEN1CARM1
SCHEMBL3553239 0.96 LMNA (0.44) LMNAHRH3KMT2AMEN1CARM1
SCHEMBL348065 0.96 HRH3 (0.50) LMNAHRH3KMT2AMEN1CARM1
SCHEMBL7007038 0.96 HRH3 (0.50) LMNAHRH3KMT2AMEN1CARM1
Hydrochloric Acid SCHEMBL10442200 0.92 HRH3 (0.47) LMNAHRH3KMT2AMEN1CARM1
Hydrochloric Acid SCHEMBL22322297 0.92 HRH3 (0.47) LMNAHRH3KMT2AMEN1CARM1
SCHEMBL3558131 0.92 HRH3 (0.47) LMNAHRH3KMT2AMEN1CARM1
SCHEMBL13776923 0.91
SCHEMBL20363777 0.89 LMNA (0.40) LMNAHRH3KMT2AMEN1CARM1
Hydrochloric Acid SCHEMBL10442465 0.89 HRH3 (0.45) LMNAHRH3KMT2AMEN1CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 209 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200283387-A1 METHOD FOR PREPARING METHIONINE ANALOGUES ADISSEO FRANCE S.A.S. (FR) 2020-09-10 US claimed
EP-3405452-A1 METHOD FOR PREPARING METHIONINE ANALOGUES Adisseo France S.A.S. (FR) 2018-11-28 EP claimed
EP-2957575-B1 OPTICALLY ACTIVE POLY(DIPHENYLACETYLENE) COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF AS OPTICAL ISOMER SEPARATING AGENT NAT UNIV CORP KANAZAWA UNIV (JP) 2017-10-18 EP claimed
WO-2017125673-A1 METHOD FOR PREPARING METHIONINE ANALOGUES ADISSEO FRANCE S.A.S. (FR) 2017-07-27 WO claimed
US-9562121-B2 Optically active poly(diphenylacetylene) compound, preparation method therefor, and use thereof as optical isomer separating agent NATIONAL UNIVERSITY CORPORATION KANAZAWA UNIVERSITY (JP) 2017-02-07 US claimed
US-20160194291-A1 STYRYL QUINAZOLINE DERIVATIVES AS PHARMACEUTICALLY ACTIVE AGENTS VICHEM CHEMIE KUTATÓ KFT. (HU) 2016-07-07 US claimed
EP-3030550-A1 STYRYL QUINAZOLINE DERIVATIVES AS PHARMACEUTICALLY ACTIVE AGENTS Vichem Chemie Kutató KFT (HU) 2016-06-15 EP claimed
US-9290592-B2 Poly(diphenylacetylene) compound, preparation method therefor, and use thereof as optical isomer separating agent NATIONAL UNIVERSITY CORPORATION KANAZAWA UNIVERSITY (JP) 2016-03-22 US claimed
US-20150376308-A1 OPTICALLY ACTIVE POLY(DIPHENYLACETYLENE) COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF AS OPTICAL ISOMER SEPARATING AGENT NATIONAL UNIVERSITY CORPORATION KANAZAWA UNIVERSITY (JP) 2015-12-31 US claimed
US-20150376309-A1 NEW POLY(DIPHENYLACETYLENE) COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF AS OPTICAL ISOMER SEPARATING AGENT National University Corporation Kanazawa University of Ishikawa ,Japan 2015-12-31 US claimed
WO-2015019121-A1 STYRYL QUINAZOLINE DERIVATIVES AS PHARMACEUTICALLY ACTIVE AGENTS VICHEM CHEMIE KUTATÓ KFT. (HU) 2015-02-12 WO claimed
EP-2091951-A2 PYRIDO[2,3-B]PYRAZINE AND[1,8]-NAPHTYRIDINE DERIVATIVES AS ALK AND C-MET INHIBITORS CEPHALON, INC. (US) 2009-08-26 EP claimed
WO-2007130468-A2 PYRIDO [2, 3-B] PYRAZINE AND [1, 8] -NAPHTHYRIDINE DERIVATIVES AS ALK AND C-MET INHIBITORS CEPHALON, INC. (US) 2007-11-15 WO claimed
CN-1213684-A Chemical Mechanical Polishing Composition CHANGXING CHEMICAL IND CO LTD (CN) 1999-04-14 CN claimed
US-5750688-A REACTING AN HALOGENATED AMINE WITH AN OXYBENZOIC ESTER; THEN A 2-(OXYPHENYL-)BENZOTHIOPHENE COMPOUND ELI LILLY AND COMPANY (US) 1998-05-12 US claimed
EP-0729956-A1 Benzothiophene compounds, intermediates, compositions, and methods ELI LILLY AND COMPANY (US) 1996-09-04 EP claimed
US-5324837-A 3,4-disubstituted-4,5-dihydro-1H-pyrazoles and a method of preparation DOWELANCO (US) 1994-06-28 US claimed
EP-0548226-A1 MONOSACCHARIDES HAVING ANTI-PROLIFERATION AND ANTI-INFLAMMATORY ACTIVITY, COMPOSITIONS AND USES THEREOF GREENWICH PHARMACEUTICALS INCORPORATED (US) 1993-06-30 EP claimed
WO-1992004359-A2 MONOSACCHARIDES HAVING ANTI-PROLIFERATION AND ANTI-INFLAMMATORY ACTIVITY, COMPOSITIONS AND USES THEREOF GREENWICH PHARMACEUTICALS, INC. (US) 1992-03-19 WO claimed
US-3985768-A Process for producing rolitetracycline E. R. SQUIBB & SONS, INC. (US) 1976-10-12 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200283387-A1 METHOD FOR PREPARING METHIONINE ANALOGUES GRM4, CHRM4, GRIA4 LMNA 3516/4885HRH3 415/4885KMT2A 1763/4885
US-20160194291-A1 STYRYL QUINAZOLINE DERIVATIVES AS PHARMACEUTICALLY ACTIVE AGENTS FLT3, BCR, STK3 LMNA 3239/4885HRH3 765/4885KMT2A 3110/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.