SCHEMBL27751680

SCHEMBL27751680

COc1cc2nccc(Nc3ccc(F)c(Cl)c3)c2cc1OC

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.70
ERBB2 P04626 2/20 0.67
KDR P35968 2/20 0.67
AURKA O14965 1/20 0.67
INSR P06213 1/20 0.67
FBP1 P09467 1/20 0.67
PDGFRB P09619 1/20 0.67
FLT4 P35916 1/20 0.67
CLK1 P49759 1/20 0.67
EPHB4 P54760 1/20 0.67
TEK Q02763 1/20 0.67
AURKB Q96GD4 1/20 0.67
SRC P12931 3/20 0.65
GAK O14976 3/20 0.62
BMPR1B O00238 1/20 0.62
EPHB6 O15197 1/20 0.62
RIPK2 O43353 1/20 0.62
ABL1 P00519 1/20 0.62
LCK P06239 1/20 0.62
EPHA1 P21709 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27751699 0.92 KDR (0.73) EGFRERBB2KDRAURKAINSR
SCHEMBL28778139 0.91 EGFR (0.60) EGFRERBB2KDRAURKAINSR
SCHEMBL31213837 0.89 EGFR (0.61) EGFRERBB2KDRAURKAINSR
SCHEMBL6352042 0.83 EGFR (0.75) EGFRERBB2KDRSRCGAK
SCHEMBL28447436 0.83 EGFR (0.66) EGFRERBB2KDRPDGFRBSRC
SCHEMBL12308286 0.83 EGFR (0.77) EGFRERBB2KDRFLT4EPHB4
SCHEMBL12484448 0.82 EGFR (0.73) EGFRERBB2KDRFBP1PDGFRB
SCHEMBL28445612 0.81 EGFR (0.68) EGFRERBB2KDRPDGFRBSRC
SCHEMBL30505605 0.81 EGFR (1.00) EGFRERBB2KDRAURKAINSR
SCHEMBL2099106 0.81 EGFR (1.00) EGFRERBB2KDRAURKAINSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101362719-B Chinolines derivates and composition containing thereof UNIV BEIJING NORMAL 2012-04-18 CN disclosed
CN-101362719-A Chinolines derivates and composition containing thereof UNIV BEIJING NORMAL (CN) 2009-02-11 CN disclosed