SCHEMBL27754979

SCHEMBL27754979

Cc1cc(-c2ccc(N)c(NC(=O)c3ccc(CN4CCOCC4)cc3)c2)ccc1S

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 8/20 0.59
RAB9A P51151 3/20 0.52
MAPK1 P28482 3/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
LMNA P02545 2/20 0.52
MAPT P10636 2/20 0.52
GALR3 O60755 1/20 0.52
HDAC3 O15379 5/20 0.51
HIF1A Q16665 6/20 0.51
EPAS1 Q99814 6/20 0.51
KCNH2 Q12809 3/20 0.51
TSHR P16473 1/20 0.49
STAT3 P40763 1/20 0.49
NPC1 O15118 1/20 0.49
HDAC2 Q92769 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4578900 0.85 HDAC1 (0.70) HDAC1RAB9AHDAC3HIF1AEPAS1
SCHEMBL4579730 0.85 HDAC1 (0.79) HDAC1RAB9AHDAC3HIF1AEPAS1
SCHEMBL4579920 0.85 HDAC1 (0.67) HDAC1RAB9AHDAC3HIF1AEPAS1
SCHEMBL14155855 0.84 RAB9A (0.60) HDAC1RAB9AMAPK1SMN1; SMN2LMNA
SCHEMBL4580174 0.83 HDAC1 (0.64) HDAC1HDAC3HIF1AEPAS1KCNH2
SCHEMBL4578211 0.83 HDAC2 (0.62) HDAC1RAB9AHDAC3HIF1AEPAS1
SCHEMBL4579854 0.82 HDAC1 (0.57) HDAC1RAB9AMAPK1SMN1; SMN2LMNA
SCHEMBL4578653 0.82 HDAC1 (0.70) HDAC1RAB9AHDAC3HIF1AEPAS1
SCHEMBL4578865 0.82 NPC1 (0.68) HDAC1RAB9AMAPK1LMNAMAPT
SCHEMBL4578145 0.80 HDAC1 (0.64) HDAC1HDAC3KCNH2HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101466670-B Inhibitors of histone deacetylase METHYLGENE INC 2013-04-17 CN claimed
CN-101466670-B Inhibitors of histone deacetylase METHYLGENE INC 2013-04-17 CN disclosed
CN-101466670-A Benzamide derivatives as inhibitors of histone deacetylase METHYLGENE INC (CA) 2009-06-24 CN disclosed