SCHEMBL27755367

SCHEMBL27755367

COCCNC(=O)c1ccc(Oc2ncnc(OC3CCN(C(=O)O)CC3)c2C)c(F)c1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 7/20 0.51
CYP2C9 P11712 2/20 0.51
PIK3CD O00329 2/20 0.44
RAB9A P51151 1/20 0.43
MET P08581 1/20 0.43
KDR P35968 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
MAPK14 Q16539 1/20 0.43
SCN9A Q15858 1/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL389132 0.90 GPR119 (0.66) GPR119CYP2C9RAB9A
SCHEMBL27747805 0.90 GPR119 (0.49) GPR119CYP2C9PIK3CDMETKDR
SCHEMBL5140735 0.87 CYP2C9 (0.44) GPR119CYP2C9METKDRMAPK14
SCHEMBL3169529 0.85 GPR119 (0.52) GPR119CYP2C9RAB9AMETKDR
SCHEMBL390219 0.85 GPR119 (0.66) GPR119CYP2C9RAB9A
SCHEMBL27755093 0.84 GPR119 (0.53) GPR119CYP2C9PIK3CD
SCHEMBL1897239 0.82 GPR119 (0.67) GPR119CYP2C9
SCHEMBL27734763 0.80 GPR119 (0.60) GPR119CYP2C9PIK3CD
SCHEMBL389599 0.80 GPR119 (0.64) GPR119CYP2C9
SCHEMBL1071546 0.80 GPR119 (0.56) GPR119CYP2C9PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101332303-A Combination therapy for the treatment of diabetes and conditions related thereto and for the treatment of conditions ameliorated by increasing a blood glp-1 level ARENA PHARM INC (US) 2008-12-31 CN disclosed