SCHEMBL27757948

SCHEMBL27757948

CCOC(=O)C(=O)OC=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.46
GLO1 Q04760 1/20 0.46
ALDH1A1 P00352 5/20 0.43
LMNA P02545 2/20 0.42
HSD17B10 Q99714 1/20 0.42
CYP2D6 P10635 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
FAAH O00519 2/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
MGAM O43451 1/20 0.40
GAA P10253 1/20 0.40
SI P14410 1/20 0.40
MGAM2 Q2M2H8 1/20 0.40
SOAT1 P35610 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
EGLN1 Q9GZT9 1/20 0.39
CYP2C9 P11712 2/20 0.38
HCAR2 Q8TDS4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7262 0.81 ALDH1A1 (0.62) NPSR1GLO1ALDH1A1LMNAHSD17B10
SCHEMBL9823358 0.81 ALDH1A1 (0.62) NPSR1GLO1ALDH1A1LMNAHSD17B10
SCHEMBL1331989 0.81 ALDH1A1 (0.62) NPSR1GLO1ALDH1A1LMNAHSD17B10
SCHEMBL27947493 0.79 ALDH1A1 (0.41) NPSR1GLO1ALDH1A1LMNAHSD17B10
SCHEMBL19958915 0.79 ALDH1A1 (0.45) NPSR1GLO1ALDH1A1LMNAHSD17B10
SCHEMBL5002228 0.78 NPSR1 (0.45) NPSR1GLO1ALDH1A1LMNAHSD17B10
SCHEMBL30076441 0.78 ALDH1A1 (0.59) NPSR1GLO1ALDH1A1LMNAHSD17B10
SCHEMBL9751764 0.78 ALDH1A1 (0.59) NPSR1GLO1ALDH1A1LMNAHSD17B10
SCHEMBL28824460 0.78 ALDH1A1 (0.59) NPSR1GLO1ALDH1A1LMNAHSD17B10
Ammonia Solution, Strong SCHEMBL12803984 0.78 ALDH1A1 (0.59) NPSR1GLO1ALDH1A1LMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101395157-A Pyrrazole derivatives as sigma receptors antagonists ESTEVE LABOR DR (ES) 2009-03-25 CN claimed
CN-109310672-A Purposes of the sigma-receptor ligand in cancer 埃斯特韦制药有限公司 2019-02-05 CN disclosed
CN-106999473-A Purposes of the sigma-receptor part in osteoarthritis 埃斯蒂文博士实验室股份有限公司 2017-08-01 CN disclosed
CN-102741248-B New (heterocycle/condense piperidines)-(piperazinyl)-1-alkane ketone or (heterocycle/condense tetramethyleneimine)-(piperazinyl)-1-alkane ketone derivatives and the purposes as p75 inhibitor thereof SAI NUOFEI (FR) 2016-01-20 CN disclosed
CN-102741248-A Novel (heterocycle/condensed piperidine)-(piperazinyl)-1-alcanone or (heterocycle/condensed pyrrolidine)-(piperazinyl)-1-alcanone derivatives, and use thereof as p75 inhibitors SANOFI AVENTIS 2012-10-17 CN disclosed
CN-102656162-A Novel (heterocycle/tetrahydropyridine)-(piperazinyl)-1-alcanone and (heterocycle/dihydropyrrolidine)-(piperazinyl)-1-alcanone derivatives, and use thereof as p75 inhibitors SANOFI SA 2012-09-05 CN disclosed
CN-102414198-A Synthesis of 3- { [ (2R) -1-methylpyrrolidin-2-yl ] methyl } -5- [2- (phenylsulfonyl) ethyl ] -1H-indole ITALIANA SINT SPA 2012-04-11 CN disclosed
CN-101395157-A Pyrrazole derivatives as sigma receptors antagonists ESTEVE LABOR DR (ES) 2009-03-25 CN disclosed