SCHEMBL27758372

SCHEMBL27758372

CC(C)(C)OC(=O)NCc1cccc(CCBr)c1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GLS O94925 11/20 0.55
KDM4A O75164 1/20 0.46
BRD4 O60885 3/20 0.46
CREBBP Q92793 1/20 0.45
AKT1 P31749 1/20 0.44
NAMPT P43490 2/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA7 P43166 1/20 0.43
CA14 Q9ULX7 1/20 0.43
NQO2 P16083 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL851272 0.89 GLS (0.55) GLSKDM4ABRD4CREBBPAKT1
SCHEMBL30192965 0.89 GLS (0.55) GLSKDM4ABRD4CREBBPAKT1
SCHEMBL21455404 0.87 GLS (0.54) GLSKDM4ABRD4CREBBPNAMPT
SCHEMBL15656811 0.86 GLS (0.53) GLSKDM4ABRD4CREBBPNAMPT
SCHEMBL5729298 0.85 GLS (0.54) GLSKDM4ABRD4CREBBPCA12
SCHEMBL16181822 0.84 GLS (0.55) GLSKDM4ABRD4CREBBPNAMPT
SCHEMBL30069429 0.84 GLS (0.55) GLSKDM4ABRD4CREBBPNAMPT
SCHEMBL1165088 0.84 GLS (0.55) GLSKDM4ABRD4CREBBPNAMPT
SCHEMBL13981921 0.84 GLS (0.55) GLSKDM4ABRD4CREBBPNAMPT
SCHEMBL8342682 0.84 GLS (0.55) GLSKDM4ABRD4CREBBPNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101691370-A Triazolo[4,5-d] pyrimidine derivatives and their use as purinergic receptor antagonists VERNALIS RES LTD 2010-04-07 CN disclosed
CN-101531631-A Substituted pyridinones as modulators of p38 map kinase PHARMACIA CORP (US) 2009-09-16 CN disclosed