SCHEMBL27760147

SCHEMBL27760147

C=CC(c1ccc(C)cc1)S(=O)(=O)n1cc(F)cc1-c1coc(C2CCCN(C(=O)c3ccc(F)cc3)C2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.42
CLPP Q16740 1/20 0.42
RAB9A P51151 1/20 0.41
ALDH1A1 P00352 3/20 0.40
LMNA P02545 2/20 0.40
TSHR P16473 2/20 0.40
HTT P42858 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPK1 P28482 2/20 0.39
MAPT P10636 1/20 0.39
ATM Q13315 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NPSR1 Q6W5P4 2/20 0.38
TP53 P04637 1/20 0.37
ALOX15 P16050 1/20 0.37
MAP3K12 Q12852 1/20 0.36
PDE2A O00408 1/20 0.36
HSD11B1 P28845 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3586168 0.85 GRM5 (0.47) GRM5CLPPRAB9AALDH1A1LMNA
SCHEMBL3586170 0.85 GRM5 (0.47) GRM5CLPPRAB9AALDH1A1LMNA
SCHEMBL3584731 0.72 GRM5 (0.68) GRM5CLPPRAB9AALDH1A1LMNA
SCHEMBL3584728 0.72 GRM5 (0.68) GRM5CLPPRAB9AALDH1A1LMNA
SCHEMBL3585860 0.71 GRM5 (0.58) GRM5CLPPRAB9ATSHRMEN1
SCHEMBL3585856 0.71 GRM5 (0.58) GRM5CLPPRAB9ATSHRMEN1
SCHEMBL3585711 0.70 GRM5 (0.57) GRM5CLPPRAB9AALDH1A1LMNA
SCHEMBL30794892 0.70 GRM5 (0.57) GRM5CLPPRAB9AALDH1A1LMNA
SCHEMBL3585701 0.70 GRM5 (0.57) GRM5CLPPRAB9AALDH1A1LMNA
SCHEMBL3586318 0.70 GRM5 (0.56) GRM5CLPPRAB9AALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101558065-A Oxazole derivatives as positive allosteric modulators of metabotropic glutamate receptors ADDEX PHARMACEUTICALS SA (CH) 2009-10-14 CN disclosed