SCHEMBL27764487

SCHEMBL27764487

O=[N+]([O-])c1cc(-c2nn[nH]n2)ccc1OCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 3/20 0.54
ABCB1 P08183 1/20 0.48
POLB P06746 1/20 0.47
XDH P47989 1/20 0.47
CTSV O60911 1/20 0.47
CTSL P07711 1/20 0.47
GP6 Q9HCN6 1/20 0.47
KDM4C Q9H3R0 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1447254 0.87 MRGPRX4 (0.44) MRGPRX4XDHKDM4C
SCHEMBL31086482 0.80 MRGPRX4 (0.56) MRGPRX4GP6KDM4C
SCHEMBL1055134 0.80 MRGPRX4 (0.56) MRGPRX4GP6KDM4C
SCHEMBL8848787 0.80 POLB (0.47) ABCB1POLBCTSVCTSL
SCHEMBL30955240 0.79 ALDH1A1 (0.67) XDH
SCHEMBL2685823 0.77 CYP11B1 (0.63) ABCB1POLBCTSVCTSL
SCHEMBL25214619 0.76 POLB (0.48) ABCB1POLBXDHCTSVCTSL
SCHEMBL30425063 0.76 POLB (0.48) ABCB1POLBXDHCTSVCTSL
SCHEMBL7116860 0.76 POLB (0.56) ABCB1POLBCTSVCTSL
SCHEMBL2685895 0.74 CYP11B1 (0.49) ABCB1POLBCTSVCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101454285-B Oxadiazole derivatives as comt inhibitors PORTELA & CA SA 2012-06-27 CN disclosed
CN-101454285-A Oxadiazole derivatives as comt inhibitors PORTELA & CA SA (PT) 2009-06-10 CN disclosed