SCHEMBL27765122

SCHEMBL27765122

COc1ccccc1-c1c(C(C)C)cnc2c(C(F)(F)F)cccc12

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 9/20 0.50
NR1H3 Q13133 9/20 0.50
ATP4A P20648 1/20 0.41
ATP4B P51164 1/20 0.41
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39
TRPA1 O75762 2/20 0.38
TRPM8 Q7Z2W7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27673874 0.85 NR1H2 (0.55) NR1H2NR1H3
SCHEMBL27653831 0.78 NR1H2 (0.43) NR1H2NR1H3ALDH1A1CYP1A2CYP3A4
SCHEMBL4012188 0.77 NR1H2 (0.63) NR1H2NR1H3
SCHEMBL27673881 0.76 NR1H2 (0.58) NR1H2NR1H3
SCHEMBL1125385 0.75 NR1H2 (0.52) NR1H2NR1H3
SCHEMBL27775437 0.74 TSHR (0.44) NR1H2AKR1C3AKR1C2ALDH1A1CYP1A2
SCHEMBL27653828 0.74 NR1H2 (0.53) NR1H2NR1H3
SCHEMBL27673864 0.72 TRPA1 (0.39) NR1H2AKR1C3AKR1C2ALDH1A1CYP1A2
SCHEMBL34599 0.72 NR1H2 (0.65) NR1H2NR1H3
SCHEMBL1125462 0.71 NR1H2 (0.53) NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN disclosed