SCHEMBL27765367

SCHEMBL27765367

COc1cc(N2CCOC[C@@H]2C)nc(-c2ccc(N)cc2)n1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ATR Q13535 16/20 0.59
PDCD1 Q15116 16/20 0.59
CD274 Q9NZQ7 16/20 0.59
CHEK1 O14757 14/20 0.59
ATRIP Q8WXE1 14/20 0.59
MTOR P42345 8/20 0.59
PIK3CA P42336 3/20 0.46
PIK3CD O00329 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3723256 0.89 PDCD1 (0.56) ATRPDCD1CD274CHEK1ATRIP
SCHEMBL3723251 0.89 PDCD1 (0.56) ATRPDCD1CD274CHEK1ATRIP
SCHEMBL20651520 0.83 PDCD1 (0.74) ATRPDCD1CD274CHEK1ATRIP
SCHEMBL20651760 0.83 PDCD1 (0.74) ATRPDCD1CD274CHEK1ATRIP
SCHEMBL3607909 0.82 PIK3CA (0.50) ATRPDCD1CD274CHEK1ATRIP
SCHEMBL27812275 0.81 MTOR (0.67) ATRPDCD1CD274CHEK1ATRIP
SCHEMBL3598683 0.81 PIK3CA (0.56) ATRPDCD1CD274CHEK1ATRIP
SCHEMBL27815303 0.81 ATR (0.49) ATRPDCD1CD274CHEK1ATRIP
SCHEMBL737810 0.80 PIK3CA (0.55) ATRPDCD1CD274CHEK1ATRIP
SCHEMBL3608383 0.80 CHEK1 (0.51) ATRPDCD1CD274CHEK1ATRIP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101541781-B Morpholino pyrimidine derivatives for the treatment of proliferative diseases ASTRAZENECA AB 2014-01-08 CN disclosed
CN-101541781-A Morpholino pyrimidine derivatives for the treatment of proliferative diseases ASTRAZENECA AB (SE) 2009-09-23 CN disclosed