SCHEMBL3723256

SCHEMBL3723256

CC1COCCN1c1cc(N2CCOCC2C)nc(-c2ccc(N)cc2)n1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 12/20 0.56
CD274 Q9NZQ7 12/20 0.56
ATR Q13535 11/20 0.56
CHEK1 O14757 10/20 0.56
ATRIP Q8WXE1 10/20 0.56
MTOR P42345 6/20 0.54
PIK3CA P42336 6/20 0.52
PIK3CD O00329 4/20 0.52
PDPK1 O15530 2/20 0.51
ROCK1 Q13464 2/20 0.51
AURKB Q96GD4 2/20 0.51
AURKA O14965 1/20 0.51
ATM Q13315 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3723251 1.00 PDCD1 (0.56) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL27765367 0.89 ATR (0.59) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL27815303 0.88 ATR (0.49) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL3598683 0.88 PIK3CA (0.56) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL737810 0.87 PIK3CA (0.55) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL27794030 0.87 CHEK1 (0.49) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL3726552 0.87 PDCD1 (0.59) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL3608383 0.87 CHEK1 (0.51) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL739897 0.85 PIK3CA (0.72) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL3607909 0.84 PIK3CA (0.50) PDCD1CD274ATRCHEK1ATRIP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010120994-A2 UREIDOARYL-AND CARBAMOYLARYL-MORPHOLINO- PYRIMIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESIS WYETH LLC (US) 2010-10-21 WO disclosed