SCHEMBL27767412

SCHEMBL27767412

NC(=O)c1cc(-c2cc(Cl)ccc2O)[nH]c1N(N)C=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 2/20 0.39
IDO1 P14902 1/20 0.38
MAPT P10636 2/20 0.38
PKM P14618 1/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
JAK2 O60674 5/20 0.36
BRD4 O60885 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
P2RX1 P51575 1/20 0.35
AR P10275 1/20 0.34
SLC9A1 P19634 1/20 0.34
MAPK1 P28482 2/20 0.34
HPN P05981 1/20 0.34
BIRC5 O15392 1/20 0.34
CDC7 O00311 1/20 0.34
PLK4 O00444 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27909732 0.89 JAK2 (0.44) PIM1MAPTJAK2BRD4KDM4E
SCHEMBL27767419 0.85 IDO1 (0.39) IDO1MAPTCA1CA2BRD4
SCHEMBL27789086 0.85 BRD4 (0.44) PIM1MAPTBRD4KDM4EALDH1A1
SCHEMBL27892770 0.81 MEN1 (0.43) JAK2BRD4ALDH1A1SLC9A1MAPK1
SCHEMBL27767424 0.80 IKBKB (0.43) MAPTJAK2BRD4KDM4ECDC7
SCHEMBL27767420 0.80 GCGR (0.40) MAPTJAK2BRD4ALDH1A1GAA
SCHEMBL27788983 0.79 PARP1 (0.44) JAK2BRD4CDC7CDK2MEN1
SCHEMBL27789042 0.77 CASP1 (0.45) JAK2BRD4ALDH1A1MAPK1CDC7
SCHEMBL27788861 0.76 BRD4 (0.41) BRD4CDC7CDK2
SCHEMBL2200770 0.74 P2RX1 (0.44) PIM1IDO1MAPTPKMCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101622229-B Pyrrole derivatives having ureido and aminocarbonyl groups as substituents SANTEN PHARMACEUTICAL CO LTD 2013-02-27 CN claimed
CN-101622229-A Novel pyrrole derivatives having ureido group and aminocarbonyl group as substituents SANTEN PHARMACEUTICAL CO LTD 2010-01-06 CN claimed
CN-101622229-B Pyrrole derivatives having ureido and aminocarbonyl groups as substituents SANTEN PHARMACEUTICAL CO LTD 2013-02-27 CN disclosed
CN-101622229-A Novel pyrrole derivatives having ureido group and aminocarbonyl group as substituents SANTEN PHARMACEUTICAL CO LTD 2010-01-06 CN disclosed