SCHEMBL27767429

SCHEMBL27767429

N#Cc1ccc(-c2cc(C(N)=O)c(N(N)C=O)[nH]2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 11/20 0.45
PARP1 P09874 3/20 0.43
CASP1 P29466 1/20 0.42
BRD4 O60885 1/20 0.39
MAP2 P11137 1/20 0.39
CCNB2 O95067 1/20 0.37
CDK1 P06493 1/20 0.37
CCNB1 P14635 1/20 0.37
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
PARP2 Q9UGN5 1/20 0.37
CHEK2 O96017 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CCNA1 P78396 1/20 0.35
MMP2 P08253 1/20 0.35
MMP3 P08254 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27788869 0.88 CDC7 (0.55) CDC7PARP1CASP1BRD4CCNA2
SCHEMBL27788861 0.85 BRD4 (0.41) CDC7PARP1BRD4CCNA2CDK2
SCHEMBL27767416 0.84 CDC7 (0.52) CDC7BRD4CCNA2CDK2CCNA1
SCHEMBL27767423 0.84 CDC7 (0.52) CDC7CASP1BRD4CCNA2CDK2
SCHEMBL27788862 0.84 BRD4 (0.56) CDC7BRD4CCNB2CDK1CCNB1
SCHEMBL27788978 0.82 BRD4 (0.39) CDC7PARP1BRD4CCNA2CDK2
SCHEMBL27788872 0.82 CHUK (0.41) CDC7PARP1BRD4CCNA2CDK2
SCHEMBL27767460 0.82 CDC7 (0.44) CDC7BRD4CCNA2CDK2CCNA1
SCHEMBL27789089 0.81 CDC7 (0.45) CDC7BRD4CHEK2CCNA2CDK2
SCHEMBL27767432 0.81 PARP10 (0.43) CDC7BRD4CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101622229-B Pyrrole derivatives having ureido and aminocarbonyl groups as substituents SANTEN PHARMACEUTICAL CO LTD 2013-02-27 CN claimed
CN-101622229-A Novel pyrrole derivatives having ureido group and aminocarbonyl group as substituents SANTEN PHARMACEUTICAL CO LTD 2010-01-06 CN claimed
CN-101622229-B Pyrrole derivatives having ureido and aminocarbonyl groups as substituents SANTEN PHARMACEUTICAL CO LTD 2013-02-27 CN disclosed
CN-101622229-A Novel pyrrole derivatives having ureido group and aminocarbonyl group as substituents SANTEN PHARMACEUTICAL CO LTD 2010-01-06 CN disclosed