SCHEMBL27768190

SCHEMBL27768190

Cc1nc2c(o1)-c1ccccc1N(C(=O)c1ccc(COC(=O)N3CCN(CCC(C)(C)C)CC3)c(C)c1)CC2

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 3/20 0.39
CD274 Q9NZQ7 3/20 0.39
AVPR2 P30518 10/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ATR Q13535 1/20 0.34
ATM Q13315 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CACNA1B Q00975 1/20 0.33
APBA1 Q02410 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27789681 0.89 PDCD1 (0.38) PDCD1CD274AVPR2ALDH1A1MAPT
SCHEMBL2704506 0.88 AVPR2 (0.44) PDCD1CD274AVPR2
SCHEMBL2705389 0.84 AVPR2 (0.42) PDCD1CD274AVPR2
SCHEMBL27789677 0.84 PDCD1 (0.38) PDCD1CD274AVPR2NPC1RAB9A
SCHEMBL2128410 0.82 AVPR2 (0.43) PDCD1CD274AVPR2
SCHEMBL18917255 0.82 AVPR2 (0.42) PDCD1CD274AVPR2
SCHEMBL27789716 0.81 PDCD1 (0.44) PDCD1CD274AVPR2
SCHEMBL2616280 0.80 PDCD1 (0.49) PDCD1CD274AVPR2NPC1RAB9A
Hydrochloric Acid SCHEMBL2129494 0.79 PDCD1 (0.48) PDCD1CD274AVPR2NPC1RAB9A
SCHEMBL2130987 0.77 AVPR2 (0.51) PDCD1CD274AVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101563347-A Vasopressin V1a antagonists VANTIA LTD (GB) 2009-10-21 CN claimed