SCHEMBL27768414

SCHEMBL27768414

c1cc2cnc3ccc(CNC4CC4)cc3n2c1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.51
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 2/20 0.49
GLA P06280 1/20 0.49
GAA P10253 1/20 0.49
HPGD P15428 1/20 0.49
HSD17B10 Q99714 1/20 0.49
HRH3 Q9Y5N1 2/20 0.38
MEN1 O00255 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38
KCNH2 Q12809 1/20 0.38
MAP4K4 O95819 4/20 0.38
PKM P14618 1/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
GRIN2B Q13224 1/20 0.34
METTL3 Q86U44 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27768404 0.95 ALDH1A1 (0.47) PARP1ALDH1A1KDM4EGLAGAA
SCHEMBL27789942 0.94 ALDH1A1 (0.46) PARP1ALDH1A1KDM4EGLAGAA
SCHEMBL27789952 0.90 PARP1 (0.51) PARP1ALDH1A1KDM4EGLAGAA
SCHEMBL27790122 0.85 ALDH1A1 (0.47) PARP1ALDH1A1KDM4EGLAGAA
SCHEMBL27789950 0.84 ALDH1A1 (0.46) PARP1ALDH1A1KDM4EGLAGAA
SCHEMBL27768387 0.82 PARP1 (0.44) PARP1ALDH1A1KDM4EGLAGAA
SCHEMBL27768407 0.81 KDM4E (0.54) PARP1ALDH1A1KDM4EGLAGAA
SCHEMBL27768388 0.80 KDM4E (0.44) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL27789949 0.80 KDM4E (0.49) PARP1ALDH1A1KDM4EGLAGAA
SCHEMBL27768390 0.75 ALDH1A1 (0.50) PARP1ALDH1A1KDM4EGLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101616919-B Poly (ADP ribose) polymerase inhibitors ABBOTT LAB 2012-10-10 CN claimed
CN-101616919-B Poly (ADP ribose) polymerase inhibitors ABBOTT LAB 2012-10-10 CN disclosed
CN-101616919-A Poly (ADP ribose) polymerase inhibitors ABBOTT LAB 2009-12-30 CN disclosed