SCHEMBL27768765

SCHEMBL27768765

CN1Cc2cc(Oc3ccc(N)cc3Cl)ccc2C1C=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.38
HTR2A P28223 1/20 0.38
PDE7A Q13946 2/20 0.37
PNLIP P16233 1/20 0.35
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
RAD52 P43351 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
SOS1 Q07889 2/20 0.32
SCN9A Q15858 1/20 0.31
MAPK14 Q16539 1/20 0.31
FFAR1 O14842 2/20 0.31
DRD2 P14416 1/20 0.31
DRD1 P21728 1/20 0.31
DRD5 P21918 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PLA2G7 Q13093 1/20 0.31
STK39 Q9UEW8 1/20 0.31
MRGPRX4 Q96LA9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27768773 0.91 HTR2A (0.38) SLC6A4HTR2APDE7APNLIPKDM4E
SCHEMBL27790238 0.83 PDE7A (0.49) PDE7AKDM4EMAPTSMN1; SMN2
SCHEMBL27936885 0.80 CA12 (0.34) HTR2AKDM4EMAPTRAD52MAPK14
SCHEMBL27768811 0.80 EZH2 (0.34) SLC6A4PDE7AKDM4EMAPTRAD52
SCHEMBL27790231 0.80 MAPT (0.33) HTR2APDE7AKDM4EMAPTRAD52
SCHEMBL28781385 0.76 PDE7A (0.39) SLC6A4HTR2APDE7APNLIPSOS1
SCHEMBL27768848 0.74 PDE7A (0.49) PDE7AKDM4EMAPTHTTSMN1; SMN2
SCHEMBL3484045 0.74 PDE7A (0.40) SLC6A4HTR2APDE7APNLIPKDM4E
SCHEMBL27948446 0.72 CA12 (0.37) HTR2AKDM4EMAPTRAD52MAPK14
SCHEMBL3485002 0.72 PDE7A (0.40) SLC6A4HTR2APDE7AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101611041-A Condensed heterocyclic compouds TAKEDA PHARMACEUTICAL (JP) 2009-12-23 CN disclosed