SCHEMBL27768920

SCHEMBL27768920

CC1(C)NC(C=O)c2ccc(Oc3ccc([N+](=O)[O-])cc3Cl)cc21

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 1/20 0.51
MEN1 O00255 7/20 0.47
KMT2A Q03164 7/20 0.47
GAA P10253 1/20 0.47
PKM P14618 1/20 0.47
KDM4E B2RXH2 1/20 0.47
HPGD P15428 3/20 0.46
ALDH1A1 P00352 10/20 0.45
MAPT P10636 7/20 0.45
LMNA P02545 5/20 0.45
SMN1; SMN2 Q16637 5/20 0.45
GPR55 Q9Y2T6 1/20 0.42
HSP90AA1 P07900 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.39
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27768921 0.82 KMT2A (0.47) PDE7AMEN1KMT2AGAAPKM
SCHEMBL27790312 0.77 PDE7A (0.52) PDE7AMEN1KMT2AGAAPKM
SCHEMBL27768770 0.77 PDE7A (0.52) PDE7AMEN1KMT2AGAAPKM
Methylamine SCHEMBL27768768 0.77 PDE7A (0.52) PDE7AMEN1KMT2AGAAPKM
SCHEMBL3484209 0.75 PDE7A (0.54) PDE7AMEN1KMT2AGAAPKM
SCHEMBL27768848 0.73 PDE7A (0.49) PDE7AMEN1KMT2AGAAPKM
SCHEMBL27790238 0.73 PDE7A (0.49) PDE7AMEN1KMT2AGAAPKM
SCHEMBL3484743 0.73 PDE7A (0.54) PDE7AMEN1KMT2AGAAPKM
SCHEMBL2529627 0.72 ALDH1A1 (0.67) PDE7AMEN1KMT2AGAAPKM
SCHEMBL3485062 0.72 PDE7A (0.56) PDE7AMEN1KMT2AGAAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101611041-A Condensed heterocyclic compouds TAKEDA PHARMACEUTICAL (JP) 2009-12-23 CN disclosed