SCHEMBL27769715

SCHEMBL27769715

Cc1cc(C(C)C(=O)C(C)c2ccc(F)c(C)c2)ccc1F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 6/20 0.53
AKR1C2 P52895 6/20 0.53
PTGS2 P35354 3/20 0.44
APP P05067 3/20 0.43
PTGS1 P23219 3/20 0.42
LMNA P02545 3/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
PSEN1 P49768 2/20 0.42
PSEN2 P49810 2/20 0.42
APH1B Q8WW43 2/20 0.42
NCSTN Q92542 2/20 0.42
APH1A Q96BI3 2/20 0.42
PSENEN Q9NZ42 2/20 0.42
FABP2 P12104 1/20 0.42
TSHR P16473 1/20 0.42
AKR1C4 P17516 1/20 0.42
ADRA2B P18089 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14465122 0.87 AKR1C3 (0.68) AKR1C3AKR1C2PTGS2APPPTGS1
SCHEMBL31240211 0.87 AKR1C3 (0.68) AKR1C3AKR1C2PTGS2APPPTGS1
SCHEMBL27711084 0.82 TDP1 (0.44) AKR1C3AKR1C2PTGS2PTGS1LMNA
SCHEMBL27852035 0.79 APP (0.42) AKR1C3AKR1C2PTGS2APPPTGS1
SCHEMBL27760488 0.79 APP (0.49) AKR1C3AKR1C2PTGS2APPPTGS1
SCHEMBL28017128 0.78 TP53 (0.45) AKR1C3AKR1C2PTGS1CYP2C9CYP2C19
SCHEMBL8251464 0.78 UGT2B7 (0.45) AKR1C3AKR1C2PTGS1LMNAMEN1
SCHEMBL8272795 0.77 AKR1C3 (0.40) AKR1C3AKR1C2PTGS2PTGS1LMNA
SCHEMBL84446 0.77 LMNA (0.52) AKR1C3AKR1C2PTGS2PTGS1LMNA
SCHEMBL18252778 0.77 AKR1C3 (0.49) AKR1C3AKR1C2PTGS2APPPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102822168-B Method for producing isoxazoline derivatives 先正达参股股份有限公司 2016-10-26 CN disclosed
CN-102822168-A Method for producing isoxazoline derivatives SYNGENTA PARTICIPATIONS AG 2012-12-12 CN disclosed
CN-101627007-A Aminoamides as orexin antagonists HOFFMANN LA ROCHE 2010-01-13 CN disclosed