SCHEMBL27770289

SCHEMBL27770289

Cc1nc(C(N)=O)sc1CCCCc1ccc(-n2cccn2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA5A P35218 1/20 0.48
CA9 Q16790 1/20 0.48
CA5B Q9Y2D0 1/20 0.48
PIK3CD O00329 4/20 0.43
PIK3CA P42336 3/20 0.43
PIK3CB P42338 3/20 0.43
PIK3CG P48736 3/20 0.43
PI4KB Q9UBF8 2/20 0.38
KLKB1 P03952 3/20 0.37
DYRK3 O43781 1/20 0.37
MAP4K4 O95819 1/20 0.37
CLK2 P49760 1/20 0.37
DYRK1A Q13627 1/20 0.37
MINK1 Q8N4C8 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
GLS O94925 1/20 0.37
SCN9A Q15858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3096972 0.78 PIK3CD (0.65) CA12CA1CA2CA5ACA9
SCHEMBL6854674 0.69 NOTUM (0.51) CHRM1LMNABRS3
SCHEMBL323044 0.69 NOTUM (0.55) MAP4K4LMNAMGLL
SCHEMBL5717609 0.68 KDM4E (0.50) CA12CA1CA2CA5ACA9
SCHEMBL28011535 0.68 PPARG (0.48) CHRM1LMNABRS3
SCHEMBL7891506 0.67 FFAR1 (0.51) LMNA
SCHEMBL1177658 0.67 NSD2 (0.57) CA12CA1CA2CA5ACA9
SCHEMBL261444 0.66 HRH2 (0.38) HRH2
SCHEMBL10029392 0.66 NOTUM (0.55) CHRM1MGLLBRS3
SCHEMBL18756509 0.66 CHRM1 (0.65) CA12CA1CA2CA5ACA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101479258-A Thiazolyl urea derivatives as phosphatidylinositol 3-kinase inhibitors NOVARTIS AG (CH) 2009-07-08 CN disclosed