Aranidipine

Aranidipine

SCHEMBL27770888

COC(=O)C1=C(C)NC(C)=C(C(=O)OCC(C)=O)C1c1ccccc1[N+](=O)[O-].[CaH2]

nearest known ligand 0.79

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 9/20 0.79
CYP2C9 P11712 9/20 0.79
ADORA3 P0DMS8 8/20 0.79
CYP3A4 P08684 8/20 0.79
CYP2C19 P33261 8/20 0.79
MAPT P10636 7/20 0.79
KMT2A Q03164 6/20 0.79
HIF1A Q16665 6/20 0.79
CACNA1C Q13936 5/20 0.79
TSHR P16473 5/20 0.79
NFKB1 P19838 5/20 0.79
LMNA P02545 4/20 0.79
CYP2D6 P10635 4/20 0.79
ABCB11 O95342 3/20 0.79
SCN1A P35498 3/20 0.79
SCN5A Q14524 3/20 0.79
SCN2A Q99250 3/20 0.79
SCN3A Q9NY46 3/20 0.79
THPO P40225 3/20 0.79
KDM4E B2RXH2 3/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Aranidipine SCHEMBL29661509 0.99 CYP1A2 (0.80) CYP1A2CYP2C9ADORA3CYP3A4CYP2C19
Aranidipine SCHEMBL49910 0.99 CYP1A2 (0.80) CYP1A2CYP2C9ADORA3CYP3A4CYP2C19
Aranidipine SCHEMBL49911 0.99 CYP1A2 (0.80) CYP1A2CYP2C9ADORA3CYP3A4CYP2C19
SCHEMBL28770057 0.90 CACNA1B (0.70) CYP1A2CYP2C9ADORA3CYP3A4CYP2C19
Nifedipine SCHEMBL8851402 0.90 ADORA3 (0.97) CYP1A2CYP2C9ADORA3CYP3A4CYP2C19
SCHEMBL5085498 0.89 ADORA3 (0.86) CYP1A2CYP2C9ADORA3CYP3A4CYP2C19
Nifedipine SCHEMBL3968 0.89 ADORA3 (1.00) CYP1A2CYP2C9ADORA3CYP3A4CYP2C19
Nifedipine SCHEMBL1172946 0.89 ADORA3 (1.00) CYP1A2CYP2C9ADORA3CYP3A4CYP2C19
Nifedipine SCHEMBL29349595 0.89 ADORA3 (1.00) CYP1A2CYP2C9ADORA3CYP3A4CYP2C19
Nifedipine SCHEMBL28674741 0.88 ADORA3 (0.93) CYP1A2CYP2C9ADORA3CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101646666-A Tricyclic compounds KYOWA HAKKO KOGYO KK JP 2010-02-10 CN disclosed