SCHEMBL27780294

SCHEMBL27780294

CC(C)(C)C(=O)ON1CCC(F)C1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 8/20 0.35
DPP8 Q6V1X1 1/20 0.35
DPP9 Q86TI2 1/20 0.35
DPP7 Q9UHL4 4/20 0.33
CTSK P43235 2/20 0.30
RIPK1 Q13546 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27664587 1.00 DPP4 (0.35) DPP4DPP8DPP9DPP7CTSK
SCHEMBL27684119 1.00 DPP4 (0.35) DPP4DPP8DPP9DPP7CTSK
SCHEMBL27713182 0.83 HRH2 (0.31)
SCHEMBL27733586 0.83 HRH2 (0.31)
SCHEMBL27720226 0.83 HRH2 (0.31)
SCHEMBL28214294 0.82 DPP4 (0.34) DPP4DPP8DPP9DPP7
SCHEMBL4698579 0.81 CHRM2 (0.36) DPP4CTSKRIPK1
SCHEMBL28265971 0.81 ALDH1A1 (0.33) DPP4DPP8DPP7CTSKRIPK1
SCHEMBL4399555 0.81 CHRM2 (0.36) DPP4CTSKRIPK1
SCHEMBL28012712 0.79

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106414435-A Amino-substituted isothiazoles 拜耳制药股份公司 2017-02-15 CN disclosed
CN-105612153-A Substituted sulfonamide compounds as TRPA1 conditioner HOFFMANN LA ROCHE 2016-05-25 CN disclosed
CN-104447707-A Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2015-03-25 CN disclosed
CN-101558059-B Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2014-12-03 CN disclosed
CN-101558059-A Hepatitis C virus inhibitors BRISTOL MYERS SQUIBB CO (US) 2009-10-14 CN disclosed