SCHEMBL27780313

SCHEMBL27780313

CC(=O)Oc1ccc2cnc(Nc3ccc(S(N)(=O)=O)cc3)nc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 6/20 0.50
KDM4E B2RXH2 1/20 0.49
CA2 P00918 7/20 0.46
CA1 P00915 6/20 0.46
CA9 Q16790 6/20 0.46
CA12 O43570 3/20 0.46
CDK1 P06493 4/20 0.45
CDK2 P24941 4/20 0.45
KDR P35968 2/20 0.45
SYK P43405 2/20 0.45
GSK3B P49841 2/20 0.45
CDC7 O00311 1/20 0.45
PLK4 O00444 1/20 0.45
CHEK1 O14757 1/20 0.45
AURKA O14965 1/20 0.45
DCLK1 O15075 1/20 0.45
PDPK1 O15530 1/20 0.45
DAPK3 O43293 1/20 0.45
JAK2 O60674 1/20 0.45
ROCK2 O75116 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27801285 0.91 IKBKB (0.50) IKBKBKDM4ECA2CA1CA9
SCHEMBL1633099 0.86 IKBKB (0.65) IKBKBCA2CA1CA9CA12
SCHEMBL1633451 0.83 CA2 (0.58) IKBKBKDM4ECA2CA1CA9
SCHEMBL1634724 0.81 IKBKB (0.62) IKBKBCA2CA1CA9CA12
SCHEMBL1570959 0.81 CDK2 (0.50) IKBKBKDM4ECA2CA1CA9
SCHEMBL1571219 0.80 IKBKB (0.48) IKBKBCA2CA1CA9CA12
SCHEMBL1631544 0.80 CDK1 (0.51) IKBKBKDM4ECA2CA1CA9
SCHEMBL1633423 0.80 IKBKB (0.63) IKBKBCA2CA1CA9CA12
SCHEMBL1633690 0.80 IKBKB (0.57) IKBKBCA2CA1CA9CA12
SCHEMBL1633518 0.80 SYK (0.53) IKBKBCA2CA1CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101652352-A Quinazolines for PDK1 inhibition NOVARTIS VACCINES & DIAGNOSTIC 2010-02-17 CN disclosed