SCHEMBL27780802

SCHEMBL27780802

N#Cc1cc(=O)n(CCN2CCC(N)CC2)c2cc(F)ccc12

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.43
DPP4 P27487 7/20 0.41
KDM1A O60341 4/20 0.40
DRD2 P14416 2/20 0.40
SLC6A4 P31645 1/20 0.40
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3840015 0.99 KCNH2 (0.42) KCNH2DPP4KDM1ADRD2SLC6A4
SCHEMBL704957 0.91 KCNH2 (0.47) KCNH2DPP4KDM1ACYP3A4CYP2D6
SCHEMBL4770655 0.85 KCNH2 (0.41) KCNH2DPP4DRD2SLC6A4HTR2A
SCHEMBL4302199 0.84 KCNH2 (0.47) KCNH2DRD2HTR2AHTR2C
SCHEMBL4303624 0.80 HTR2C (0.43) DRD2SLC6A4HTR2AHTR2C
SCHEMBL4302247 0.79 KCNA3 (0.49) KCNH2DPP4DRD2
SCHEMBL705731 0.78 KCNH2 (0.40) KCNH2DRD2SLC6A4HTR2AHTR2C
SCHEMBL705950 0.78 SCN7A (0.43) KCNH2KDM1A
SCHEMBL706822 0.78 KCNH2 (0.43) KCNH2DRD2SLC6A4
Hydrochloric Acid SCHEMBL3870194 0.77 KCNH2 (0.43) KCNH2DRD2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101516889-B Derivatives and analogs of n-ethylquinolones and n-ethylazaquinolones GLAXO GROUP LTD 2013-07-31 CN disclosed
CN-101516889-A Derivatives and analogs of n-ethylquinolones and n-ethylazaquinolones GLAXO GROUP LTD (GB) 2009-08-26 CN disclosed