SCHEMBL27780914

SCHEMBL27780914

CC(C(=O)C(C)c1ccnc(Cl)c1)c1ccnc(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMARCA2 P51531 7/20 0.41
SMARCA4 P51532 6/20 0.41
RECQL P46063 1/20 0.40
FFAR2 O15552 1/20 0.38
OPRM1 P35372 1/20 0.37
OPRK1 P41145 1/20 0.37
KCNH2 Q12809 1/20 0.37
RIOK2 Q9BVS4 1/20 0.37
KDM4C Q9H3R0 1/20 0.36
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
LOX P28300 1/20 0.36
LOXL3 P58215 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.36
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2183698 0.87 AKR1C3 (0.44) RECQLAKR1C3AKR1C2
SCHEMBL29272210 0.83 PTGS1 (0.47) SMARCA2SMARCA4FFAR2OPRM1OPRK1
SCHEMBL13332664 0.80 GPR119 (0.44) SMARCA2SMARCA4RECQLAKR1C3AKR1C2
SCHEMBL1979197 0.80 GPR119 (0.44) SMARCA2SMARCA4RECQLAKR1C3AKR1C2
SCHEMBL27924260 0.79 PSEN1 (0.44) SMARCA2SMARCA4
SCHEMBL2040052 0.79 RECQL (0.44) SMARCA2SMARCA4RECQLFFAR2OPRM1
SCHEMBL30003916 0.79 RECQL (0.44) SMARCA2SMARCA4RECQLFFAR2OPRM1
SCHEMBL4330263 0.79 RECQL (0.44) SMARCA2SMARCA4RECQLFFAR2OPRM1
SCHEMBL2759112 0.78 RECQL (0.42) SMARCA2SMARCA4RECQLFFAR2OPRM1
SCHEMBL27845906 0.78 KDM1A (0.37) RIOK2AKR1C3AKR1C2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101627007-A Aminoamides as orexin antagonists HOFFMANN LA ROCHE 2010-01-13 CN disclosed
CN-101516874-A Pyrrole derivatives for the treatment of cytokine mediated diseases NOVARTIS AG (CH) 2009-08-26 CN disclosed