SCHEMBL27782868

SCHEMBL27782868

O=C(Nc1nc(CCc2ccccc2)cs1)c1ccccc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 3/20 0.74
KDM4E B2RXH2 2/20 0.66
PDE5A O76074 2/20 0.66
NPC1 O15118 3/20 0.59
RAB9A P51151 3/20 0.59
SRC P12931 1/20 0.58
CASP3 P42574 1/20 0.58
SENP7 Q9BQF6 1/20 0.58
SENP6 Q9GZR1 1/20 0.58
SMN1; SMN2 Q16637 2/20 0.56
PDE1A P54750 1/20 0.55
PDE1B Q01064 1/20 0.55
PDE1C Q14123 1/20 0.55
SCD O00767 3/20 0.55
KDM4A O75164 1/20 0.54
KDM4B O94953 1/20 0.54
ADORA3 P0DMS8 1/20 0.54
KDM5B Q9UGL1 1/20 0.54
CDK5 Q00535 2/20 0.54
CDK5R1 Q15078 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4874993 0.91 AOC3 (0.74) AOC3KDM4EPDE5ANPC1RAB9A
SCHEMBL13679462 0.86 AOC3 (0.70) AOC3KDM4EPDE5ANPC1RAB9A
SCHEMBL4874675 0.85 AOC3 (0.63) AOC3KDM4EPDE5ANPC1RAB9A
Hydrochloric Acid SCHEMBL4875657 0.85 AOC3 (0.71) AOC3KDM4EPDE5ANPC1RAB9A
SCHEMBL8430108 0.84 AOC3 (0.76) AOC3NPC1RAB9ASMN1; SMN2
SCHEMBL91391 0.83 KDM4E (0.69) AOC3KDM4EPDE5ANPC1RAB9A
SCHEMBL27599948 0.83 KDM4E (0.78) AOC3KDM4EPDE5ANPC1RAB9A
SCHEMBL2227204 0.83 KDM4E (0.69) AOC3KDM4EPDE5ANPC1RAB9A
SCHEMBL2664517 0.83 KDM4E (0.69) AOC3KDM4EPDE5ANPC1RAB9A
Carbamic Acid SCHEMBL4874681 0.82 AOC3 (0.67) AOC3KDM4EPDE5ASCDCDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101747327-A Aromatic amide thiazole derivative, preparation method and application thereof UNIV BEIJING 2010-06-23 CN claimed
CN-101747327-B Aromatic amide thiazole derivative, preparation method and application thereof UNIV BEIJING 2013-03-27 CN disclosed
CN-101747327-A Aromatic amide thiazole derivative, preparation method and application thereof UNIV BEIJING 2010-06-23 CN disclosed